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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50251486   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Dual specificity tyrosine-phosphorylation-regulated kinase 1A


(Homo sapiens (Human))		BDBM50251486
PNG
(CHEMBL4066607)
Show SMILES c1[nH]c2cnccc2c1-c1ccnc2ccccc12
Show InChI InChI=1S/C16H11N3/c1-2-4-15-12(3-1)11(6-8-18-15)14-9-19-16-10-17-7-5-13(14)16/h1-10,19H
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MMDB

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Article
PubMed
n/an/a 277n/an/an/an/an/an/a



Rigel Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...

Bioorg Med Chem Lett 27: 2617-2621 (2017)


Article DOI: 10.1016/j.bmcl.2017.03.037
BindingDB Entry DOI: 10.7270/Q2SN0CFP
More data for this
Ligand-Target Pair