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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50453920   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Potassium voltage-gated channel subfamily H member 2


(Homo sapiens (Human))		BDBM50453920
PNG
(CHEMBL4217431)
Show SMILES Cl.Cl.FCCOc1cccc(CCN2CCN(CCc3ccccc3)CC2)c1
Show InChI InChI=1S/C22H29FN2O/c23-11-18-26-22-8-4-7-21(19-22)10-13-25-16-14-24(15-17-25)12-9-20-5-2-1-3-6-20/h1-8,19H,9-18H2
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MMDB

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PC cid
PC sid
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Article
PubMed
n/an/a 4.31E+3n/an/an/an/an/an/a



University of Kentucky

Curated by ChEMBL


Assay Description
Displacement of [3H]Dofetilide from human ERG expressed in HEK293 cells after 60 mins by scintillation spectrometry

Bioorg Med Chem Lett 27: 5467-5472 (2017)


Article DOI: 10.1016/j.bmcl.2017.10.039
BindingDB Entry DOI: 10.7270/Q2BP05B5
More data for this
Ligand-Target Pair