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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50455583   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Protein kinase C iota type


(Homo sapiens (Human))		BDBM50455583
PNG
(CHEMBL4204387)
Show SMILES Cn1cnc2ccc(cc12)-c1ccnc2[nH]ccc12
Show InChI InChI=1S/C15H12N4/c1-19-9-18-13-3-2-10(8-14(13)19)11-4-6-16-15-12(11)5-7-17-15/h2-9H,1H3,(H,16,17)
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 2.00E+4n/an/an/an/an/an/a



Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL


Assay Description
Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...

J Med Chem 61: 4386-4396 (2018)


Article DOI: 10.1021/acs.jmedchem.8b00060
BindingDB Entry DOI: 10.7270/Q2V69N5Z
More data for this
Ligand-Target Pair