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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50496798   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Bromodomain-containing protein 4


(Homo sapiens (Human))		BDBM50496798
PNG
(CHEMBL3220849)
Show SMILES Cc1noc(C)c1-c1ccc2n(Cc3ccc(O)cc3)c(C)nc2c1
Show InChI InChI=1S/C20H19N3O2/c1-12-20(13(2)25-22-12)16-6-9-19-18(10-16)21-14(3)23(19)11-15-4-7-17(24)8-5-15/h4-10,24H,11H2,1-3H3
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 2.00E+3n/an/an/an/an/an/a



University of Oxford

Curated by ChEMBL


Assay Description
Inhibition of BRD4 bromodomain-1 (unknown origin) by AlphaScreen assay

Medchemcomm 4: 140-144 (2013)


Article DOI: 10.1039/c2md20189e
BindingDB Entry DOI: 10.7270/Q2RX9G1D
More data for this
Ligand-Target Pair