Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
CDK-activating kinase assembly factor MAT1 (Homo sapiens (Human)) | BDBM59227 (Pyrazolopyrimidone analog, RGB-286147) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 71 | n/a | n/a | n/a | n/a | n/a | n/a |
GPC Biotech, Inc. | Assay Description Inhibition of in vitro kinase activity of purified CDKs. | Chem Biol 12: 1103-15 (2005) Article DOI: 10.1016/j.chembiol.2005.08.008 BindingDB Entry DOI: 10.7270/Q28W3BR6 | |||||||||||
More data for this Ligand-Target Pair |