Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
C-X-C chemokine receptor type 6 (Mus musculus) | BDBM50539457 (CHEMBL4645971) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanford Burnham Prebys Medical Discovery Institute Curated by ChEMBL | Assay Description Antagonist activity at mouse CXCR6 by DiscoveRx cell based beta-arrestin assay | Bioorg Med Chem Lett 30: (2020) Article DOI: 10.1016/j.bmcl.2019.126899 BindingDB Entry DOI: 10.7270/Q2K077T6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 6 (Mus musculus) | BDBM50539483 (CHEMBL4637126) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >4.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanford Burnham Prebys Medical Discovery Institute Curated by ChEMBL | Assay Description Antagonist activity at mouse CXCR6 by DiscoveRx cell based beta-arrestin assay | Bioorg Med Chem Lett 30: (2020) Article DOI: 10.1016/j.bmcl.2019.126899 BindingDB Entry DOI: 10.7270/Q2K077T6 | |||||||||||
More data for this Ligand-Target Pair |