Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Ghrelin O-acyltransferase (Mus musculus) | BDBM50548065 (CHEMBL4785875) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of mouse GOAT expressed in baculovirus infected sf9 insect cell microsomes using biotinylated des-acyl ghrelin and octanoyl-CoA -CoA as su... | Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Mus musculus) | BDBM50548066 (CHEMBL4791105) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of mouse GOAT expressed in baculovirus infected sf9 insect cell microsomes using biotinylated des-acyl ghrelin and octanoyl-CoA -CoA as su... | Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Mus musculus) | BDBM50548069 (CHEMBL4741670) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co... | Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Mus musculus) | BDBM50548072 (CHEMBL4778987) | UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co... | Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Mus musculus) | BDBM50548074 (CHEMBL4750990) | UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co... | Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Mus musculus) | BDBM50548068 (CHEMBL4753228) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using ghrelin(1 to 5) pentapeptide as substrate preincub... | Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Mus musculus) | BDBM50548067 (CHEMBL4762372) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using ghrelin(1 to 5) pentapeptide as substrate preincub... | Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Mus musculus) | BDBM50548073 (CHEMBL4756686) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co... | Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Mus musculus) | BDBM50548070 (CHEMBL4784392) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co... | Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ghrelin O-acyltransferase (Mus musculus) | BDBM50548071 (CHEMBL4788110) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of N-terminal His10-tagged mouse GOAT expressed in baculovirus infected sf9 insect cell membrane using proghrelin-His8 and [3H]octanoyl Co... | Citation and Details Article DOI: 10.1039/d0md00210k BindingDB Entry DOI: 10.7270/Q2KS6W53 | |||||||||||
More data for this Ligand-Target Pair |