Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
DNA polymerase III PolC-type (Staphylococcus aureus) | BDBM50177653 (5-allyl-6-chloro-2-(2,3-dihydro-1H-inden-5-ylamino...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Targanta Therapeutics Inc. Curated by ChEMBL | Assay Description Inhibition of DNA polymerase3C from Staphylococcus aureus | Bioorg Med Chem Lett 16: 891-6 (2006) Article DOI: 10.1016/j.bmcl.2005.11.009 BindingDB Entry DOI: 10.7270/Q2125S75 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA polymerase III PolC-type (Staphylococcus aureus) | BDBM50177648 (2-(2,3-dihydro-1H-inden-5-ylamino)-6-hydroxy-5-(3-...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Targanta Therapeutics Inc. Curated by ChEMBL | Assay Description Inhibition of DNA polymerase3C from Staphylococcus aureus | Bioorg Med Chem Lett 16: 891-6 (2006) Article DOI: 10.1016/j.bmcl.2005.11.009 BindingDB Entry DOI: 10.7270/Q2125S75 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA polymerase III PolC-type (Staphylococcus aureus) | BDBM50177644 (2-(2,3-dihydro-1H-inden-5-ylamino)-6-hydroxy-5-(3-...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Targanta Therapeutics Inc. Curated by ChEMBL | Assay Description Inhibition of DNA polymerase3C from Staphylococcus aureus | Bioorg Med Chem Lett 16: 891-6 (2006) Article DOI: 10.1016/j.bmcl.2005.11.009 BindingDB Entry DOI: 10.7270/Q2125S75 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA polymerase III PolC-type (Staphylococcus aureus) | BDBM50177654 (4-(3-(2-(2,3-dihydro-1H-inden-5-ylamino)-4-hydroxy...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Targanta Therapeutics Inc. Curated by ChEMBL | Assay Description Inhibition of DNA polymerase3C from Staphylococcus aureus | Bioorg Med Chem Lett 16: 891-6 (2006) Article DOI: 10.1016/j.bmcl.2005.11.009 BindingDB Entry DOI: 10.7270/Q2125S75 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA polymerase III PolC-type (Staphylococcus aureus) | BDBM50177645 (2-(2,3-dihydro-1H-inden-5-ylamino)-6-hydroxy-5-(3-...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Targanta Therapeutics Inc. Curated by ChEMBL | Assay Description Inhibition of DNA polymerase3C from Staphylococcus aureus | Bioorg Med Chem Lett 16: 891-6 (2006) Article DOI: 10.1016/j.bmcl.2005.11.009 BindingDB Entry DOI: 10.7270/Q2125S75 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA polymerase III PolC-type (Staphylococcus aureus) | BDBM50177651 (5-benzyl-2-(3-ethyl-4-methylphenylamino)-6-hydroxy...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Targanta Therapeutics Inc. Curated by ChEMBL | Assay Description Inhibition of DNA polymerase3C from Staphylococcus aureus | Bioorg Med Chem Lett 16: 891-6 (2006) Article DOI: 10.1016/j.bmcl.2005.11.009 BindingDB Entry DOI: 10.7270/Q2125S75 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA polymerase III PolC-type (Staphylococcus aureus) | BDBM50177657 (2-(2,3-dihydro-1H-inden-5-ylamino)-6-hydroxy-5-(3-...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Targanta Therapeutics Inc. Curated by ChEMBL | Assay Description Inhibition of DNA polymerase3C from Staphylococcus aureus | Bioorg Med Chem Lett 16: 891-6 (2006) Article DOI: 10.1016/j.bmcl.2005.11.009 BindingDB Entry DOI: 10.7270/Q2125S75 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA polymerase III PolC-type (Staphylococcus aureus) | BDBM50177647 (4-(3-(2-(2,3-dihydro-1H-inden-5-ylamino)-4-hydroxy...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Targanta Therapeutics Inc. Curated by ChEMBL | Assay Description Inhibition of DNA polymerase3C from Staphylococcus aureus | Bioorg Med Chem Lett 16: 891-6 (2006) Article DOI: 10.1016/j.bmcl.2005.11.009 BindingDB Entry DOI: 10.7270/Q2125S75 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA polymerase III PolC-type (Staphylococcus aureus) | BDBM50177665 (5-allyl-2-(3-ethyl-4-methylphenylamino)-6-hydroxyp...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Targanta Therapeutics Inc. Curated by ChEMBL | Assay Description Inhibition of DNA polymerase3C from Staphylococcus aureus | Bioorg Med Chem Lett 16: 891-6 (2006) Article DOI: 10.1016/j.bmcl.2005.11.009 BindingDB Entry DOI: 10.7270/Q2125S75 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA polymerase III PolC-type (Staphylococcus aureus) | BDBM50177656 (5-(3-(4-aminophenoxy)propyl)-2-(2,3-dihydro-1H-ind...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Targanta Therapeutics Inc. Curated by ChEMBL | Assay Description Inhibition of DNA polymerase3C from Staphylococcus aureus | Bioorg Med Chem Lett 16: 891-6 (2006) Article DOI: 10.1016/j.bmcl.2005.11.009 BindingDB Entry DOI: 10.7270/Q2125S75 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA polymerase III PolC-type (Staphylococcus aureus) | BDBM50177660 (2-(2,3-dihydro-1H-inden-5-ylamino)-6-hydroxy-5-(3-...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.16E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Targanta Therapeutics Inc. Curated by ChEMBL | Assay Description Inhibition of DNA polymerase3C from Staphylococcus aureus | Bioorg Med Chem Lett 16: 891-6 (2006) Article DOI: 10.1016/j.bmcl.2005.11.009 BindingDB Entry DOI: 10.7270/Q2125S75 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA polymerase III PolC-type (Staphylococcus aureus) | BDBM50177652 (2-(2,3-dihydro-1H-inden-5-ylamino)-6-hydroxy-5-(4-...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Targanta Therapeutics Inc. Curated by ChEMBL | Assay Description Inhibition of DNA polymerase3C from Staphylococcus aureus | Bioorg Med Chem Lett 16: 891-6 (2006) Article DOI: 10.1016/j.bmcl.2005.11.009 BindingDB Entry DOI: 10.7270/Q2125S75 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA polymerase III PolC-type (Staphylococcus aureus) | BDBM50177646 (5-(but-3-enyl)-2-(2,3-dihydro-1H-inden-5-ylamino)-...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.79E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Targanta Therapeutics Inc. Curated by ChEMBL | Assay Description Inhibition of DNA polymerase3C from Staphylococcus aureus | Bioorg Med Chem Lett 16: 891-6 (2006) Article DOI: 10.1016/j.bmcl.2005.11.009 BindingDB Entry DOI: 10.7270/Q2125S75 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA polymerase III PolC-type (Staphylococcus aureus) | BDBM50177663 (2-(2,3-dihydro-1H-inden-5-ylamino)-6-hydroxy-5-phe...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Targanta Therapeutics Inc. Curated by ChEMBL | Assay Description Inhibition of DNA polymerase3C from Staphylococcus aureus | Bioorg Med Chem Lett 16: 891-6 (2006) Article DOI: 10.1016/j.bmcl.2005.11.009 BindingDB Entry DOI: 10.7270/Q2125S75 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA polymerase III PolC-type (Staphylococcus aureus) | BDBM50177659 (5-allyl-2-(2,3-dihydro-1H-inden-5-ylamino)-6-hydro...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Targanta Therapeutics Inc. Curated by ChEMBL | Assay Description Inhibition of DNA polymerase3C from Staphylococcus aureus | Bioorg Med Chem Lett 16: 891-6 (2006) Article DOI: 10.1016/j.bmcl.2005.11.009 BindingDB Entry DOI: 10.7270/Q2125S75 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA polymerase III PolC-type (Staphylococcus aureus) | BDBM50177655 (5-benzyl-2-(2,3-dihydro-1H-inden-5-ylamino)-6-hydr...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Targanta Therapeutics Inc. Curated by ChEMBL | Assay Description Inhibition of DNA polymerase3C from Staphylococcus aureus | Bioorg Med Chem Lett 16: 891-6 (2006) Article DOI: 10.1016/j.bmcl.2005.11.009 BindingDB Entry DOI: 10.7270/Q2125S75 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA polymerase III PolC-type (Staphylococcus aureus) | BDBM50177658 (6-amino-2-(3-ethyl-4-methylphenylamino)pyrimidin-4...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.04E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Targanta Therapeutics Inc. Curated by ChEMBL | Assay Description Inhibition of DNA polymerase3C from Staphylococcus aureus | Bioorg Med Chem Lett 16: 891-6 (2006) Article DOI: 10.1016/j.bmcl.2005.11.009 BindingDB Entry DOI: 10.7270/Q2125S75 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DNA polymerase III PolC-type (Staphylococcus aureus) | BDBM50177649 (5-allyl-6-amino-2-(3-ethyl-4-methylphenylamino)pyr...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.64E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Targanta Therapeutics Inc. Curated by ChEMBL | Assay Description Inhibition of DNA polymerase3C from Staphylococcus aureus | Bioorg Med Chem Lett 16: 891-6 (2006) Article DOI: 10.1016/j.bmcl.2005.11.009 BindingDB Entry DOI: 10.7270/Q2125S75 | |||||||||||
More data for this Ligand-Target Pair |