Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556715![]() (CHEMBL4782344) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid UniChem | n/a | n/a | 630 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Assay Description In vitro inhibitory activity against beta-2 adrenergic receptor was measured by the inhibition of isoproterenol-induced relaxation of PGF2-alpha cont... | Citation and Details | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556717![]() (CHEMBL4780703) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 630 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556698![]() (CHEMBL2375494) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 650 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556698![]() (CHEMBL2375494) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | n/a | n/a | 650 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Assay Description In vitro inhibitory activity against beta-2 adrenergic receptor was measured by the inhibition of isoproterenol-induced relaxation of PGF2-alpha cont... | Citation and Details | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556715![]() (CHEMBL4782344) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 880 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556716![]() (CHEMBL4796964) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 910 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556721![]() (CHEMBL4790746) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.01E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556719![]() (CHEMBL4782590) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.08E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556710![]() (CHEMBL4741257) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.23E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556706![]() (CHEMBL4797370) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.49E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556718![]() (CHEMBL4787771) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.52E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556699![]() (CHEMBL4746541) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.64E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556705![]() (CHEMBL4793323) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.72E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556708![]() (CHEMBL4795327) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.76E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556700![]() (CHEMBL4761208) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.81E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556722![]() (CHEMBL4791780) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.81E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556720![]() (CHEMBL4745132) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.82E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556709![]() (CHEMBL4783011) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.37E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556703![]() (CHEMBL4761078) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.57E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556701![]() (CHEMBL4746014) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.63E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556702![]() (CHEMBL4763588) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.82E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556704![]() (CHEMBL4740701) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.02E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556713![]() (CHEMBL4748854) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.29E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556714![]() (CHEMBL4777734) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.54E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556707![]() (CHEMBL4762863) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.87E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556723![]() (CHEMBL240484) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.45E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556723![]() (CHEMBL240484) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid UniChem | n/a | n/a | 5.45E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Assay Description In vitro inhibitory activity against beta-2 adrenergic receptor was measured by the inhibition of isoproterenol-induced relaxation of PGF2-alpha cont... | Citation and Details | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556712![]() (CHEMBL4798117) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.64E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50556711![]() (CHEMBL4755423) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.13E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01133 BindingDB Entry DOI: 10.7270/Q27P9327 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G-protein coupled receptor 52 (Homo sapiens (Human)) | BDBM50405604![]() (CHEMBL5279049) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Assay Description In vitro inhibitory activity against beta-2 adrenergic receptor was measured by the inhibition of isoproterenol-induced relaxation of PGF2-alpha cont... | Citation and Details | |||||||||||
More data for this Ligand-Target Pair |