Compile Data Set for Download or QSAR

Found 7 hits of ic50 for UniProtKB: P14672   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Solute carrier family 2, facilitated glucose transporter member 4 (Homo sapiens)	BDBM50277370 (CHEMBL4171968) Show SMILES COc1ccc(cc1)C(=O)N(Cc1ccncc1)Cc1cccc(OCCc2ccc(F)cc2)c1 Show InChI InChI=1S/C29H27FN2O3/c1-34-27-11-7-25(8-12-27)29(33)32(20-23-13-16-31-17-14-23)21-24-3-2-4-28(19-24)35-18-15-22-5-9-26(30)10-6-22/h2-14,16-17,19H,15,18,20-21H2,1H3	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.70E+3	n/a	n/a	n/a	n/a	n/a	n/a
Emory University Curated by ChEMBL					Assay Description Antagonist activity at human GLUT4 expressed in HEK293 cells transfected with GLUT1 shRNA assessed as inhibition of [3H]2-deoxy-D-glucose uptake prei...				Eur J Med Chem 139: 573-586 (2017) Article DOI: 10.1016/j.ejmech.2017.08.029 BindingDB Entry DOI: 10.7270/Q2NC63Q7
					More data for this Ligand-Target Pair
Solute carrier family 2, facilitated glucose transporter member 4 (Homo sapiens)	BDBM50565143 (CHEMBL4793560) Show SMILES O=C(CN1C(=O)S\C(=C\c2ccco2)C1=O)Nc1nc2ccccc2s1 Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem	Article PubMed	n/a	n/a	6.80E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of transport activity of human GLUT4 expressed in hexose transporter deficient W4000fgy1 erg4 yeast cells assessed as reduction in transpo...				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112603 BindingDB Entry DOI: 10.7270/Q25Q50T2
					More data for this Ligand-Target Pair
Solute carrier family 2, facilitated glucose transporter member 4 (Homo sapiens)	BDBM50277369 (CHEMBL4160688) Show SMILES COc1ccc(cc1)C(=O)N(Cc1ccncc1)Cc1cccc(OCc2cccc(OC)c2)c1 Show InChI InChI=1S/C29H28N2O4/c1-33-26-11-9-25(10-12-26)29(32)31(19-22-13-15-30-16-14-22)20-23-5-3-8-28(17-23)35-21-24-6-4-7-27(18-24)34-2/h3-18H,19-21H2,1-2H3	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem Patents	Article PubMed	n/a	n/a	1.10E+4	n/a	n/a	n/a	n/a	n/a	n/a
Emory University Curated by ChEMBL					Assay Description Antagonist activity at human GLUT4 expressed in HEK293 cells transfected with GLUT1 shRNA assessed as inhibition of [3H]2-deoxy-D-glucose uptake prei...				Eur J Med Chem 139: 573-586 (2017) Article DOI: 10.1016/j.ejmech.2017.08.029 BindingDB Entry DOI: 10.7270/Q2NC63Q7
					More data for this Ligand-Target Pair
Solute carrier family 2, facilitated glucose transporter member 4 (Homo sapiens)	BDBM50277373 (CHEMBL4165190) Show SMILES COc1ccc(CC(=O)N(Cc2ccncc2)Cc2cccc(OCCc3ccc(F)cc3)c2)cc1 Show InChI InChI=1S/C30H29FN2O3/c1-35-28-11-7-24(8-12-28)20-30(34)33(21-25-13-16-32-17-14-25)22-26-3-2-4-29(19-26)36-18-15-23-5-9-27(31)10-6-23/h2-14,16-17,19H,15,18,20-22H2,1H3	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.82E+4	n/a	n/a	n/a	n/a	n/a	n/a
Emory University Curated by ChEMBL					Assay Description Antagonist activity at human GLUT4 expressed in HEK293 cells transfected with GLUT1 shRNA assessed as inhibition of [3H]2-deoxy-D-glucose uptake prei...				Eur J Med Chem 139: 573-586 (2017) Article DOI: 10.1016/j.ejmech.2017.08.029 BindingDB Entry DOI: 10.7270/Q2NC63Q7
					More data for this Ligand-Target Pair
Solute carrier family 2, facilitated glucose transporter member 4 (Homo sapiens)	BDBM50277387 (CHEMBL4164091) Show SMILES Oc1cccc(CNCc2ccncc2)c1 Show InChI InChI=1S/C13H14N2O/c16-13-3-1-2-12(8-13)10-15-9-11-4-6-14-7-5-11/h1-8,15-16H,9-10H2	PDB UniProtKB/SwissProt GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Emory University Curated by ChEMBL					Assay Description Antagonist activity at human GLUT4 expressed in HEK293 cells transfected with GLUT1 shRNA assessed as inhibition of [3H]2-deoxy-D-glucose uptake prei...				Eur J Med Chem 139: 573-586 (2017) Article DOI: 10.1016/j.ejmech.2017.08.029 BindingDB Entry DOI: 10.7270/Q2NC63Q7
					More data for this Ligand-Target Pair
Solute carrier family 2, facilitated glucose transporter member 4 (Homo sapiens)	BDBM50565142 (CHEMBL4776246) Show SMILES Cc1cccc2sc(NC(=O)CN3C(=O)S\C(=C\c4ccco4)C3=O)nc12 Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.23E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of transport activity of human GLUT4 expressed in hexose transporter deficient W4000fgy1 erg4 yeast cells assessed as reduction in transpo...				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112603 BindingDB Entry DOI: 10.7270/Q25Q50T2
					More data for this Ligand-Target Pair
Solute carrier family 2, facilitated glucose transporter member 4 (Homo sapiens)	BDBM50565144 (CHEMBL4786111) Show SMILES Clc1ccc(NC(=O)CN2C(=O)S\C(=C\c3ccco3)C2=O)cc1Cl Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.52E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of transport activity of human GLUT4 expressed in hexose transporter deficient W4000fgy1 erg4 yeast cells assessed as reduction in transpo...				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112603 BindingDB Entry DOI: 10.7270/Q25Q50T2
					More data for this Ligand-Target Pair