Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Apolipoprotein(a) (Human) | BDBM544449 ((2S)-3-[3-[[Bis[[3-[(2S)-2-carboxy-2-[(3R)-pyrroli...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <0.314 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The in vitro binding affinity of compounds to the intended target human Apo(a) protein is tested in a competitive binding assay. Human Apo(a) protein... | Citation and Details BindingDB Entry DOI: 10.7270/Q21N84BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apolipoprotein(a) (Human) | BDBM544455 (3-[3-[[bis[[3-[2-carboxy-2-[(3R)-pyrrolidin-3-yl]p...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <0.314 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The in vitro binding affinity of compounds to the intended target human Apo(a) protein is tested in a competitive binding assay. Human Apo(a) protein... | Citation and Details BindingDB Entry DOI: 10.7270/Q21N84BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apolipoprotein(a) (Human) | BDBM544456 ((2S)-3-[3-[3-[(2S)-2-Carboxy-2-[(3R)-pyrrolidin-3-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <0.314 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The in vitro binding affinity of compounds to the intended target human Apo(a) protein is tested in a competitive binding assay. Human Apo(a) protein... | Citation and Details BindingDB Entry DOI: 10.7270/Q21N84BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apolipoprotein(a) (Human) | BDBM544454 ((2S)-3-[3-[[[3-[(2S)-2-Carboxy-2-[(3R)-pyrrolidin-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.13 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The in vitro binding affinity of compounds to the intended target human Apo(a) protein is tested in a competitive binding assay. Human Apo(a) protein... | Citation and Details BindingDB Entry DOI: 10.7270/Q21N84BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apolipoprotein(a) (Human) | BDBM544458 ((2R)-3-Phenyl-2-[(3S)-pyrrolidin-3-yl]propanoic ac...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 126 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The in vitro binding affinity of compounds to the intended target human Apo(a) protein is tested in a competitive binding assay. Human Apo(a) protein... | Citation and Details BindingDB Entry DOI: 10.7270/Q21N84BN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apolipoprotein(a) (Human) | BDBM544457 ((2S)-3-Phenyl-2-[(3R)-pyrrolidin-3-yl]propanoic ac...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 152 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The in vitro binding affinity of compounds to the intended target human Apo(a) protein is tested in a competitive binding assay. Human Apo(a) protein... | Citation and Details BindingDB Entry DOI: 10.7270/Q21N84BN | |||||||||||
More data for this Ligand-Target Pair |