Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50002243 (1-Cyclopropylmethyl-4-(4-nitro-phenoxymethyl)-pipe...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ANSTO Curated by ChEMBL | Assay Description Receptor binding affinity against Sigma receptor | J Med Chem 40: 1657-67 (1997) Article DOI: 10.1021/jm960720+ BindingDB Entry DOI: 10.7270/Q29G5KX8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Mus musculus (Mouse)) | BDBM50002243 (1-Cyclopropylmethyl-4-(4-nitro-phenoxymethyl)-pipe...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Du Pont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro binding affinity for the mouse sigma opioid receptor | J Med Chem 35: 4344-61 (1992) BindingDB Entry DOI: 10.7270/Q28P614G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 2A/2B/2C (Mus musculus (Mouse)) | BDBM50002243 (1-Cyclopropylmethyl-4-(4-nitro-phenoxymethyl)-pipe...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 215 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Du Pont Merck Pharmaceutical Company Curated by ChEMBL | Assay Description In vitro binding affinity for serotonin 5-hydroxytryptamine (5-HT) 2 receptors | J Med Chem 35: 4344-61 (1992) BindingDB Entry DOI: 10.7270/Q28P614G | |||||||||||
More data for this Ligand-Target Pair |