Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Vasopressin V1a receptor (Homo sapiens (Human)) | BDBM50079261 (CHEMBL3416768) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 48 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Teikyo University Curated by ChEMBL | Assay Description Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V1a receptor transfected in CHO cell membranes | J Med Chem 58: 3268-73 (2015) Article DOI: 10.1021/acs.jmedchem.5b00289 BindingDB Entry DOI: 10.7270/Q21R6S7F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vasopressin V2 receptor (Homo sapiens (Human)) | BDBM50079261 (CHEMBL3416768) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 880 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Teikyo University Curated by ChEMBL | Assay Description Displacement of [3H]-(Arg8)-vasopressin from human vasopressin V2 receptor transfected in CHO cell membranes | J Med Chem 58: 3268-73 (2015) Article DOI: 10.1021/acs.jmedchem.5b00289 BindingDB Entry DOI: 10.7270/Q21R6S7F | |||||||||||
More data for this Ligand-Target Pair |