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Compile Data Set for Download or QSAR

Found 1 hit of ki for monomerid = 50091394   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Histamine H3 receptor


(Rattus norvegicus (rat))		BDBM50091394
PNG
(1-{4-[3-(1H-Imidazol-4-yl)-propoxy]-phenyl}-ethano...)
Show SMILES C\C(=N/OCc1ccccc1)c1ccc(OCCCc2cnc[nH]2)cc1
Show InChI InChI=1S/C21H23N3O2/c1-17(24-26-15-18-6-3-2-4-7-18)19-9-11-21(12-10-19)25-13-5-8-20-14-22-16-23-20/h2-4,6-7,9-12,14,16H,5,8,13,15H2,1H3,(H,22,23)/b24-17+
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PubMed
 24n/an/an/an/an/an/an/an/a



Freie Universität Berlin

Curated by ChEMBL


Assay Description
Histamine H3 receptor antagonist activity in an assay with K+ evoked depolarization-induced release of [3H]-histamine from rat synaptosomes.

J Med Chem 43: 3335-43 (2000)


BindingDB Entry DOI: 10.7270/Q2RR1XGV
More data for this
Ligand-Target Pair