Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Solute carrier family 2, facilitated glucose transporter member 4 (Rattus norvegicus) | BDBM50277375 (CHEMBL4173323) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | 2.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Antagonist activity at GLUT4 in rat adipocytes assessed as reduction in insulin-stimulated [3H]2-deoxyglucose uptake preincubated for 1 min followed ... | Eur J Med Chem 139: 573-586 (2017) Article DOI: 10.1016/j.ejmech.2017.08.029 BindingDB Entry DOI: 10.7270/Q2NC63Q7 | |||||||||||
More data for this Ligand-Target Pair |