Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465543 (CHEMBL4278778) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetry | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair |