Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Steroidogenic factor 1 (Homo sapiens (Human)) | BDBM50511469![]() (CHEMBL4515639) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Binding affinity to SF1 LBD (218 to 461 residues) (unknown origin) expressed in Escherichia coli BL21 pLysS measured after overnight incubation by fl... | ACS Med Chem Lett 11: 365-370 (2020) Article DOI: 10.1021/acsmedchemlett.9b00442 BindingDB Entry DOI: 10.7270/Q2K35Z0D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Steroidogenic factor 1 (Homo sapiens (Human)) | BDBM50418303![]() (CHEMBL1765959) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a |
Emory University Curated by ChEMBL | Assay Description Binding affinity to human SF1 LBD (218 to 461 residues) expressed in Escherichia coli BL21 by electrophoretic mobility shift assay | ACS Med Chem Lett 11: 365-370 (2020) Article DOI: 10.1021/acsmedchemlett.9b00442 BindingDB Entry DOI: 10.7270/Q2K35Z0D | |||||||||||
More data for this Ligand-Target Pair |