Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Protein AF-9 (Homo sapiens) | BDBM50459744 (CHEMBL4204744) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University Curated by ChEMBL | Assay Description Binding affinity to MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) by Bio-layer interferometry | ACS Med Chem Lett 9: 895-900 (2018) Article DOI: 10.1021/acsmedchemlett.8b00175 BindingDB Entry DOI: 10.7270/Q2DV1NHX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein AF-9 (Homo sapiens) | BDBM50576674 (CHEMBL4850575) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 370 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to AF9 YEATS domain (1 to 138 residues) (unknown origin) by isothermal titration calorimetry | Citation and Details Article DOI: 10.1016/j.bmc.2021.116342 BindingDB Entry DOI: 10.7270/Q2BZ69W1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein AF-9 (Homo sapiens) | BDBM50576675 (CHEMBL4848627) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to AF9 YEATS domain (1 to 138 residues) (unknown origin) by isothermal titration calorimetry | Citation and Details Article DOI: 10.1016/j.bmc.2021.116342 BindingDB Entry DOI: 10.7270/Q2BZ69W1 | |||||||||||
More data for this Ligand-Target Pair |