Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
cAMP-dependent protein kinase type I-alpha regulatory subunit [R243A] (Homo sapiens (Human)) | BDBM218808 (8-[Fluo]-cAMP) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 7.29 | n/a | n/a | n/a | n/a | n/a |
University of California, San Diego | Assay Description The ability of the R subunit basic patch mutants to bind cAMP in the absence of the C subunit was tested using the fluorescent cAMP analogue, 8-[fluo... | Biochemistry 56: 1536-1545 (2017) Article DOI: 10.1021/acs.biochem.6b01152 BindingDB Entry DOI: 10.7270/Q2DJ5DHF | |||||||||||
More data for this Ligand-Target Pair |