Compile Data Set for Download or QSAR

Found 64 hits Enz. Inhib. hit(s) with all data for entry = 10507   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542437 (1-[4-(4-fluorophenyl)-2-pyrazol-1-yl-cyclopentyl] ...) Show SMILES NC1CCCN(C1)C1CC(CC1n1cccn1)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2.80	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542002 (1-[4-(4-fluorophenyl)-2-(triazol-2-yl)cyclopentyl]...) Show SMILES NC1CCCN(C1)C1CC(CC1n1nccn1)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	3.37	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542439 (5-fluoro-1-[4-(4-fluorophenyl)-2-pyrazol-1-yl-cycl...) Show SMILES NC1CC(F)CN(C1)C1CC(CC1n1cccn1)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	3.40	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542462 (5-fluoro-1-[4-(4-fluorophenyl)-2-pyrimidin-4-yloxy...) Show SMILES NC1CC(F)CN(C1)C1CC(CC1Oc1ccncn1)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	3.44	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542462 (5-fluoro-1-[4-(4-fluorophenyl)-2-pyrimidin-4-yloxy...) Show SMILES NC1CC(F)CN(C1)C1CC(CC1Oc1ccncn1)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	3.68	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542143 (1-[2-(3-amino-1-piperidyl)-4-(4-fluorophenyl)cyclo...) Show SMILES NC1CCCN(C1)C1CC(CC1n1cc(nn1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	3.78	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542444 (5-fluoro-1-[4-(4-fluorophenyl)-2-(tetrazol-2-yl) c...) Show SMILES NC1CC(F)CN(C1)C1CC(CC1n1ncnn1)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	4.03	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542199 (1-[2-(3-amino-5-fluoro-1-piperidyl)-4-(4-fluorophe...) Show SMILES NC1CC(F)CN(C1)C1CC(CC1n1cc(cn1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	4.06	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542143 (1-[2-(3-amino-1-piperidyl)-4-(4-fluorophenyl)cyclo...) Show SMILES NC1CCCN(C1)C1CC(CC1n1cc(nn1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	4.28	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542121 (1-[2-(3-amino-1-piperidyl)-4-(4-fluorophenyl)cyclo...) Show SMILES NC1CCCN(C1)C1CC(CC1n1ccc(c1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	5.31	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542121 (1-[2-(3-amino-1-piperidyl)-4-(4-fluorophenyl)cyclo...) Show SMILES NC1CCCN(C1)C1CC(CC1n1ccc(c1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	5.39	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542199 (1-[2-(3-amino-5-fluoro-1-piperidyl)-4-(4-fluorophe...) Show SMILES NC1CC(F)CN(C1)C1CC(CC1n1cc(cn1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	6.22	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542456 (1-[2-(4-chloropyridazin-3-yl)oxy-4-(4-fluorophenyl...) Show SMILES NC1CCCN(C1)C1CC(CC1Oc1nnccc1Cl)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	6.56	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542439 (5-fluoro-1-[4-(4-fluorophenyl)-2-pyrazol-1-yl-cycl...) Show SMILES NC1CC(F)CN(C1)C1CC(CC1n1cccn1)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	6.64	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542446 (1-[2-(3-amino-1-piperidyl)-4-(4-fluorophenyl)cyclo...) Show SMILES NC1CCCN(C1)C1CC(CC1n1cnc(n1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	7.10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542457 (6-[2-(3-amino-5-fluoro-1-piperidyl)-4-(4-fluorophe...) Show SMILES NC1CC(F)CN(C1)C1CC(CC1Oc1ccc(nn1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	7.20	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542445 (1-[4-(4-fluorophenyl)-2-(tetrazol-2-yl)cyclopentyl...) Show SMILES NC1CCCN(C1)C1CC(CC1n1ncnn1)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	7.55	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542111 (1-[2-(3-amino-1-piperidyl)-4-(4-fluorophenyl)cyclo...) Show SMILES NC1CCCN(C1)C1CC(CC1n1cc(cn1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	7.97	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542437 (1-[4-(4-fluorophenyl)-2-pyrazol-1-yl-cyclopentyl] ...) Show SMILES NC1CCCN(C1)C1CC(CC1n1cccn1)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	7.97	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542111 (1-[2-(3-amino-1-piperidyl)-4-(4-fluorophenyl)cyclo...) Show SMILES NC1CCCN(C1)C1CC(CC1n1cc(cn1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	8.31	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542448 (4-[2-(3-amino-1-piperidyl)-4-(4-fluoro-3-methoxy-p...) Show SMILES COc1cc(ccc1F)C1CC(Oc2ccc(cc2)C#N)C(C1)N1CCCC(N)C1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	9.51	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542459 (6-[2-(3-amino-1-piperidyl)-4-(4-fluorophenyl) cycl...) Show SMILES N[C@@H]1CCCN(C1)C1CC(CC1Oc1ccc(cn1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	9.51	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542458 (US11274091, Example 25 | l-[4-(4-fluorophenyl)-2-(...) Show SMILES NC1CCCN(C1)C1CC(CC1Oc1cc(F)cnn1)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	9.93	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542444 (5-fluoro-1-[4-(4-fluorophenyl)-2-(tetrazol-2-yl) c...) Show SMILES NC1CC(F)CN(C1)C1CC(CC1n1ncnn1)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	10.6	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542465 (5-[2-(3-amino-1-piperidyl)-4-(4-fluorophenyl) cycl...) Show SMILES NC1CCCN(C1)C1CC(CC1Oc1cnc(nc1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	10.6	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542456 (1-[2-(4-chloropyridazin-3-yl)oxy-4-(4-fluorophenyl...) Show SMILES NC1CCCN(C1)C1CC(CC1Oc1nnccc1Cl)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	11.3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542463 (2-[2-(3-amino-1-piperidyl)-4-(4-fluorophenyl) cycl...) Show SMILES NC1CCCN(C1)C1CC(CC1Oc1ncc(cn1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	11.5	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542457 (6-[2-(3-amino-5-fluoro-1-piperidyl)-4-(4-fluorophe...) Show SMILES NC1CC(F)CN(C1)C1CC(CC1Oc1ccc(nn1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	>11.8	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542464 (5-[2-(3-amino-1-piperidyl)-4-(4-fluorophenyl) cycl...) Show SMILES NC1CCCN(C1)C1CC(CC1Oc1cnc(cn1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	13.7	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542453 (2-[2-(3-amino-1-piperidyl)-4-phenyl-cyclopentoxy] ...) Show SMILES NC1CCCN(C1)C1CC(CC1Oc1ccccc1C#N)c1ccccc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	14.1	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542446 (1-[2-(3-amino-1-piperidyl)-4-(4-fluorophenyl)cyclo...) Show SMILES NC1CCCN(C1)C1CC(CC1n1cnc(n1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	14.3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542443 (5-fluoro-1-[4-(4-fluorophenyl)-2-(1,2,4-triazol-1-...) Show SMILES N[C@@H]1C[C@@H](F)CN(C1)[C@@H]1C[C@@H](C[C@H]1n1cncn1)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem	US Patent	n/a	n/a	16	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542201 (1-[2-(3-amino-4,4-difluoro-1-piperidyl)-4-(4-fluor...) Show SMILES NC1CN(CCC1(F)F)C1CC(CC1n1cc(cn1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	16.2	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542447 (4-[2-(3-amino-1-piperidyl)-4-(4-fluoro-3-hydroxy-p...) Show SMILES NC1CCCN(C1)C1CC(CC1Oc1ccc(cc1)C#N)c1ccc(F)c(O)c1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	17.4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542454 (4-[2-(3-amino-1-piperidyl)-4-phenyl-cyclopentoxy]-...) Show SMILES NC1CCCN(C1)C1CC(CC1Oc1ccc(cc1Cl)C#N)c1ccccc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	17.4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542201 (1-[2-(3-amino-4,4-difluoro-1-piperidyl)-4-(4-fluor...) Show SMILES NC1CN(CCC1(F)F)C1CC(CC1n1cc(cn1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	17.5	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542002 (1-[4-(4-fluorophenyl)-2-(triazol-2-yl)cyclopentyl]...) Show SMILES NC1CCCN(C1)C1CC(CC1n1nccn1)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	17.7	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542461 (1-[4-(4-fluorophenyl)-2-pyridazin-3-yloxy-cyclopen...) Show SMILES NC1CCCN(C1)C1CC(CC1Oc1cccnn1)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	17.8	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542449 (4-[2-(3-amino-1-piperidyl)-4-(3-fluorophenyl) cycl...) Show SMILES NC1CCCN(C1)C1CC(CC1Oc1ccc(cc1Cl)C#N)c1cccc(F)c1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	19.3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542119 (1-[2-(3-amino-1-piperidyl)-4-(4-fluorophenyl)cyclo...) Show SMILES NC1CCCN(C1)C1CC(CC1n1ccc(n1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<19.9	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542450 (4-[2-(3-amino-4,4-difluoro-1-piperidyl)-4-(4-fluor...) Show SMILES NC1CN(CCC1(F)F)C1CC(CC1Oc1ccc(cc1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	20.7	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542460 (6-[2-(3-amino-1-piperidyl)-4-(4-fluorophenyl) cycl...) Show SMILES NC1CCCN(C1)C1CC(CC1Oc1ccc(cn1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	22	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542448 (4-[2-(3-amino-1-piperidyl)-4-(4-fluoro-3-methoxy-p...) Show SMILES COc1cc(ccc1F)C1CC(Oc2ccc(cc2)C#N)C(C1)N1CCCC(N)C1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	22.5	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542463 (2-[2-(3-amino-1-piperidyl)-4-(4-fluorophenyl) cycl...) Show SMILES NC1CCCN(C1)C1CC(CC1Oc1ncc(cn1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	24	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542452 (4-[2-(3-amino-1-piperidyl)-4-(4-fluorophenyl) cycl...) Show SMILES NC1CCCN(C1)C1CC(CC1Oc1ccc(C#N)c(F)c1)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	25.1	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542459 (6-[2-(3-amino-1-piperidyl)-4-(4-fluorophenyl) cycl...) Show SMILES N[C@@H]1CCCN(C1)C1CC(CC1Oc1ccc(cn1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	25.5	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 3 (Homo sapiens (Human))	BDBM542464 (5-[2-(3-amino-1-piperidyl)-4-(4-fluorophenyl) cycl...) Show SMILES NC1CCCN(C1)C1CC(CC1Oc1cnc(cn1)C#N)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	25.5	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542445 (1-[4-(4-fluorophenyl)-2-(tetrazol-2-yl)cyclopentyl...) Show SMILES NC1CCCN(C1)C1CC(CC1n1ncnn1)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	26.7	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542455 (6-[2-(3-amino-5-fluoro-1-piperidyl)-4-(4-fluorophe...) Show SMILES Cc1cc(nnc1OC1CC(CC1N1CC(N)CC(F)C1)c1ccc(F)cc1)C#N Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	28.8	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair
Short transient receptor potential channel 6 (Homo sapiens (Human))	BDBM542443 (5-fluoro-1-[4-(4-fluorophenyl)-2-(1,2,4-triazol-1-...) Show SMILES N[C@@H]1C[C@@H](F)CN(C1)[C@@H]1C[C@@H](C[C@H]1n1cncn1)c1ccc(F)cc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem	US Patent	n/a	n/a	29.8	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description For TRPC6 current recording, the intracellular solution contained (in mM): 120 CsOH, 120 Aspartate, 20 CsCl, 2 MgCl2, 0.4 CaCl2, 10 HEPES, 2 Na2ATP, ...				Citation and Details BindingDB Entry DOI: 10.7270/Q27D2ZBR
					More data for this Ligand-Target Pair

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