Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM478990 ((R)-1-(5-(3-((5-chloropyrimidin-2- yl)amino)pyrrol...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of compounds was determined using one protein kinase in a customized, thiol free assay. IC50 values were measured by testing 10 conc... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479012 ((R)-N-(4-(3-((5-chloro-4- methylpyrimidin-2- yl)am...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of compounds was determined using one protein kinase in a customized, thiol free assay. IC50 values were measured by testing 10 conc... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479014 ((R)-N-(4-(3-((5-chloro-4- methoxypyridin-2- yl)ami...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479014 ((R)-N-(4-(3-((5-chloro-4- methoxypyridin-2- yl)ami...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of compounds was determined using one protein kinase in a customized, thiol free assay. IC50 values were measured by testing 10 conc... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479015 ((R)-N-(4-(3-((5-chloro-4- methylpyridin-2- yl)amin...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of compounds was determined using one protein kinase in a customized, thiol free assay. IC50 values were measured by testing 10 conc... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM478981 ((R)-N-(4-(3-((5-chloro-4- cyclopropoxypyrimidin-2-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of compounds was determined using one protein kinase in a customized, thiol free assay. IC50 values were measured by testing 10 conc... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479018 ((R)-N-(4-(3-((5- cyclopropylpyrimidin-2- yl)amino)...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of compounds was determined using one protein kinase in a customized, thiol free assay. IC50 values were measured by testing 10 conc... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479022 ((R)-N-(4-(3-((5-chloro-4- (methylamino)pyrimidin-2...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479022 ((R)-N-(4-(3-((5-chloro-4- (methylamino)pyrimidin-2...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of compounds was determined using one protein kinase in a customized, thiol free assay. IC50 values were measured by testing 10 conc... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM478963 ((R)-1-(6-(3-((5-chloro-4- methoxypyrimidin-2- yl)a...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of compounds was determined using one protein kinase in a customized, thiol free assay. IC50 values were measured by testing 10 conc... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM478965 ((R)-N-(2-chloro-4-(3-((5-chloro-4- methoxypyrimidi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of compounds was determined using one protein kinase in a customized, thiol free assay. IC50 values were measured by testing 10 conc... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM478967 ((R)-N-(4-(3-((5-chloro-4- methoxypyrimidin-2- yl)a...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of compounds was determined using one protein kinase in a customized, thiol free assay. IC50 values were measured by testing 10 conc... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM478970 ((R)-N-(4-(3-((5-chloro-4- methoxypyrimidin-2- yl)a...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of compounds was determined using one protein kinase in a customized, thiol free assay. IC50 values were measured by testing 10 conc... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM478966 ((R)-N-(2-chloro-4-(3-((5- chloropyrimidin-2- yl)am...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of compounds was determined using one protein kinase in a customized, thiol free assay. IC50 values were measured by testing 10 conc... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM478971 ((R)-N-(4-(3-((5-chloro-4- methoxypyrimidin-2- yl)a...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of compounds was determined using one protein kinase in a customized, thiol free assay. IC50 values were measured by testing 10 conc... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479036 ((R)-N-(4-(3-((5-bromopyrimidin-2- yl)amino)pyrroli...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of compounds was determined using one protein kinase in a customized, thiol free assay. IC50 values were measured by testing 10 conc... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479038 ((R)-N-(4-(3-((5-chloro-4- methoxypyrimidin-2- yl)a...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of compounds was determined using one protein kinase in a customized, thiol free assay. IC50 values were measured by testing 10 conc... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479039 ((R)-N-(2-methyl-4-(3-((5- (trifluoromethyl)pyrimid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of compounds was determined using one protein kinase in a customized, thiol free assay. IC50 values were measured by testing 10 conc... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479046 ((R)-N-(4-(3-((5-chloro-4- (dimethylamino)pyrimidin...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479048 ((R)-N-(4-(3-((5-chloro-4-(2- methoxyethoxy)pyrimid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479050 ((R)-N-(4-(3-((4-amino-5- chloropyrimidin-2- yl)ami...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479051 ((R)-N-(4-(3-((4-amino-5- (trifluoromethyl)pyrimidi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479052 ((R)-N-(4-(3-((5-chloro-4- (trifluoromethyl)pyrimid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479007 ((R)-N-(4-(3-((5-chloro-4- methoxypyrimidin-2- yl)a...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479055 ((R)-N-(4-(3-((5-chloro-4- phenoxypyrimidin-2- yl)a...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479056 ((R)-N-(4-(3-((5-chloro-4- ethoxypyrimidin-2- yl)am...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479062 ((R)-N-(4-(3-((5-chloro-4-(2- cyanoethoxy)pyrimidin...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479064 ((R)-N-(4-(3-((5-bromopyrimidin-2- yl)amino)pyrroli...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479022 ((R)-N-(4-(3-((5-chloro-4- (methylamino)pyrimidin-2...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479080 ((R)-N-(4-(3-((4-(methylamino)-5- (trifluoromethyl)...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479084 ((R)-N-(4-(3-((5-chloro-4- methoxypyrimidin-2- yl)a...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479085 ((R)-N-(4-(3-((5-chloropyrimidin-2- yl)amino)pyrrol...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479097 ((R)-N-(4-(3-((5-chloro-4-(2- hydroxyethoxy)pyrimid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479007 ((R)-N-(4-(3-((5-chloro-4- methoxypyrimidin-2- yl)a...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479046 ((R)-N-(4-(3-((5-chloro-4- (dimethylamino)pyrimidin...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479103 (N-(4-((R)-3-((5-chloro-4- ethoxypyrimidin-2- yl)am...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479104 ((R)-N-(4-(3-((5-chloro-4- ethoxypyrimidin-2- yl)am...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479111 ((R)-N-(4-(3-((5-chloro-4- methoxypyrimidin-2- yl)a...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479112 ((R)-N-(6-(3-((5-chloro-4- ethoxypyrimidin-2- yl)am...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479084 ((R)-N-(4-(3-((5-chloro-4- methoxypyrimidin-2- yl)a...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479117 ((R)-N-(4-(3-((5-bromopyrimidin-2- yl)amino)pyrroli...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479122 (N-(4-((R)-3-((5-bromopyrimidin-2- yl)amino)pyrroli...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479123 (N-(4-((R)-3-((5-bromopyrimidin-2- yl)amino)pyrroli...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479124 ((R)-N-(4-(3-((5-cyano-4- methoxypyrimidin-2- yl)am...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479126 ((E)-N-(4-((R)-3-((5-chloro-4- methoxypyrimidin-2- ...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479128 ((E)-N-(4-((R)-3-((5-chloro-4- methoxypyrimidin-2- ...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479139 (N-(4-((2S,4R)-4-((5-chloro-4- methoxypyrimidin-2-y...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479140 ((R)-N-(4-(3-((5-ethynylpyrimidin-2- yl)amino)pyrro...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479141 ((R)-N-(4-(3-((5-ethynyl-4- methoxypyrimidin-2- yl)...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM479142 (N-(4-((2R,4R)-4-((5-chloro-4- methoxypyrimidin-2-y...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The IC50 profile of test compounds was determined using three protein kinases. IC50 values were measured by testing 10 concentrations (1×10−04M... | Citation and Details BindingDB Entry DOI: 10.7270/Q2R78JFB | |||||||||||
More data for this Ligand-Target Pair |
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