Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM397500 (US9994525, Example 15) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University | Assay Description Receptor binding assays were performed in at least 5 concentrations, with two parallel samples in each concentrations, in at least two independent ex... | Bioorg Med Chem 17: 2461-75 (2009) BindingDB Entry DOI: 10.7270/Q2RN3B6Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM397499 (US9994525, Example 14) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University | Assay Description Receptor binding assays were performed in at least 5 concentrations, with two parallel samples in each concentrations, in at least two independent ex... | Bioorg Med Chem 17: 2461-75 (2009) BindingDB Entry DOI: 10.7270/Q2RN3B6Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM397498 (US9994525, Example 13) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University | Assay Description Receptor binding assays were performed in at least 5 concentrations, with two parallel samples in each concentrations, in at least two independent ex... | Bioorg Med Chem 17: 2461-75 (2009) BindingDB Entry DOI: 10.7270/Q2RN3B6Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM397497 (US9994525, Example 12) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University | Assay Description Receptor binding assays were performed in at least 5 concentrations, with two parallel samples in each concentrations, in at least two independent ex... | Bioorg Med Chem 17: 2461-75 (2009) BindingDB Entry DOI: 10.7270/Q2RN3B6Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM397501 (US9994525, Example 16) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University | Assay Description Receptor binding assays were performed in at least 5 concentrations, with two parallel samples in each concentrations, in at least two independent ex... | Bioorg Med Chem 17: 2461-75 (2009) BindingDB Entry DOI: 10.7270/Q2RN3B6Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM397495 (US9994525, Example 10) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University | Assay Description Receptor binding assays were performed in at least 5 concentrations, with two parallel samples in each concentrations, in at least two independent ex... | Bioorg Med Chem 17: 2461-75 (2009) BindingDB Entry DOI: 10.7270/Q2RN3B6Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM397487 (US9994525, Example 3) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University | Assay Description Receptor binding assays were performed in at least 5 concentrations, with two parallel samples in each concentrations, in at least two independent ex... | Bioorg Med Chem 17: 2461-75 (2009) BindingDB Entry DOI: 10.7270/Q2RN3B6Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM397490 (US9994525, Example 5) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University | Assay Description Receptor binding assays were performed in at least 5 concentrations, with two parallel samples in each concentrations, in at least two independent ex... | Bioorg Med Chem 17: 2461-75 (2009) BindingDB Entry DOI: 10.7270/Q2RN3B6Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM397496 (US9994525, Example 11) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University | Assay Description Receptor binding assays were performed in at least 5 concentrations, with two parallel samples in each concentrations, in at least two independent ex... | Bioorg Med Chem 17: 2461-75 (2009) BindingDB Entry DOI: 10.7270/Q2RN3B6Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM397494 (US9994525, Example 9) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University | Assay Description Receptor binding assays were performed in at least 5 concentrations, with two parallel samples in each concentrations, in at least two independent ex... | Bioorg Med Chem 17: 2461-75 (2009) BindingDB Entry DOI: 10.7270/Q2RN3B6Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM397493 (US9994525, Example 8) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University | Assay Description Receptor binding assays were performed in at least 5 concentrations, with two parallel samples in each concentrations, in at least two independent ex... | Bioorg Med Chem 17: 2461-75 (2009) BindingDB Entry DOI: 10.7270/Q2RN3B6Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM397492 (US9994525, Example 7) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University | Assay Description Receptor binding assays were performed in at least 5 concentrations, with two parallel samples in each concentrations, in at least two independent ex... | Bioorg Med Chem 17: 2461-75 (2009) BindingDB Entry DOI: 10.7270/Q2RN3B6Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM397491 (US9994525, Example 6) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University | Assay Description Receptor binding assays were performed in at least 5 concentrations, with two parallel samples in each concentrations, in at least two independent ex... | Bioorg Med Chem 17: 2461-75 (2009) BindingDB Entry DOI: 10.7270/Q2RN3B6Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM397489 (US9994525, Example 4) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University | Assay Description Receptor binding assays were performed in at least 5 concentrations, with two parallel samples in each concentrations, in at least two independent ex... | Bioorg Med Chem 17: 2461-75 (2009) BindingDB Entry DOI: 10.7270/Q2RN3B6Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM397475 (US9994525, Example 1) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University | Assay Description Receptor binding assays were performed in at least 5 concentrations, with two parallel samples in each concentrations, in at least two independent ex... | Bioorg Med Chem 17: 2461-75 (2009) BindingDB Entry DOI: 10.7270/Q2RN3B6Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM397476 (US9994525, Example 2) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's University | Assay Description Receptor binding assays were performed in at least 5 concentrations, with two parallel samples in each concentrations, in at least two independent ex... | Bioorg Med Chem 17: 2461-75 (2009) BindingDB Entry DOI: 10.7270/Q2RN3B6Z | |||||||||||
More data for this Ligand-Target Pair |