Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43207![]() (2-[(2,6-dichlorobenzyl)amino]-3-methyl-butyric aci...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | PCBioAssay | n/a | n/a | n/a | n/a | 5.37E+3 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43220![]() (4-[3-(4-methoxyphenyl)-5-phenyl-3,4-dihydropyrazol...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 704 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43253![]() (MLS000119085 | N-(2-methylphenyl)-1-(8-quinolinyls...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 3.45E+3 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43211![]() (6-(4-Methoxy-phenyl)-2-piperazin-1-yl-pyrimidine-4...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem | PCBioAssay | n/a | n/a | n/a | n/a | 3.09E+4 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43212![]() ((5Z)-5-[(2Z)-2-(1-ethyl-3,3-dimethyl-2-indolyliden...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 5.42E+3 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43254![]() ((1Z)-1-[(benzylamino)methylene]-3-nitro-6,7,8,9-te...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 4.02E+3 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43216![]() ((5Z)-2-(3,4-dihydro-1H-isoquinolin-2-yl)-5-(4-etho...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 3.59E+4 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43255![]() (1-(3,6-dichloro-9-carbazolyl)-3-[2-(3H-indol-3-yl)...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 2.63E+4 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43256![]() (7-(3,4-dihydro-1H-isoquinolin-2-ylcarbonyl)-3-(2-m...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem | PCBioAssay | n/a | n/a | n/a | n/a | 851 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43250![]() (MLS000680398 | N-[3-[1-esyl-5-(p-tolyl)-2-pyrazoli...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 2.67E+3 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43257![]() (2-[2-(benzenesulfonyl)-5-(4-methylphenyl)-3,4-dihy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 1.69E+3 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43258![]() (2-[(3S,3'aR,8'aS,8'bS)-5,7-dimethyl-1',2,3'-trioxo...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 1.99E+3 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43259![]() (MLS000621545 | N-({[4-({[amino(imino)methyl]amino}...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 738 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43220![]() (4-[3-(4-methoxyphenyl)-5-phenyl-3,4-dihydropyrazol...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 704 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43221![]() (2-(benzoylcarbamothioylamino)-5,5-dimethyl-4,7-dih...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 171 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43223![]() (2-(2,3,5,6-tetramethylbenzoyl)benzoic acid | 2-(2,...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 6.26E+3 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43230![]() (2-(7,8-dihydro-6H-cyclopenta[2,3]thieno[2,4-d]pyri...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 2.76E+3 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43231![]() ((E)-3-(1-benzyl-3-thiophen-2-ylpyrazol-4-yl)prop-2...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem | PCBioAssay | n/a | n/a | n/a | n/a | 3.64E+3 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43233![]() (1-benzyl-5-chloro-3-methyl-pyrazole-4-carboxylic a...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 4.88E+3 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43235![]() (2-[2-(4-chlorophenyl)ethylamino]benzoic acid | UNM...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem | PCBioAssay | n/a | n/a | n/a | n/a | 741 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43241![]() (1-[2-(2,5-dimethylphenoxy)ethyl]-3-indolecarboxyli...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 158 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM43221![]() (2-(benzoylcarbamothioylamino)-5,5-dimethyl-4,7-dih...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 171 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A (Canis lupus familiaris) | BDBM42384![]() (2-(2-phenylethylsulfanyl)pyridine-3-carboxylic aci...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | n/a | n/a | 358 | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2T15221 | |||||||||||
More data for this Ligand-Target Pair |