Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449838![]() (CHEMBL3718273) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.66E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449886![]() (CHEMBL4163593) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.36E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449840![]() (CHEMBL3716462) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.06E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449841![]() (CHEMBL3716488) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 5.29E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449842![]() (CHEMBL3719295) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.36E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449843![]() (CHEMBL3718813) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 9.40E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449844![]() (CHEMBL3717553) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 334 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449845![]() (CHEMBL3717211) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 188 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449846![]() (CHEMBL3715235) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 52 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449847![]() (CHEMBL3715097) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.74E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449848![]() (CHEMBL3717178) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.18E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449849![]() (CHEMBL3717089) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 265 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449850![]() (CHEMBL3718541) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 471 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449851![]() (CHEMBL3716581) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 7.47E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449852![]() (CHEMBL3716540) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 747 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449853![]() (CHEMBL4162685) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.74E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449854![]() (CHEMBL3715203) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.67E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449855![]() (CHEMBL3715105) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.97E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449856![]() (CHEMBL3715743) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 747 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449857![]() (CHEMBL3715539) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4.71E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449858![]() (CHEMBL3717389) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 188 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449859![]() (CHEMBL3718400) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 67 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449860![]() (CHEMBL3716980) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 94 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449861![]() (CHEMBL3715081) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 47 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50010261![]() ((3R,4aR,5S,6S,6aS,10S,10aR,10bS)-3-ethenyl-6,10,10...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 47 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449862![]() (CHEMBL1479446) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.88E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449863![]() (CHEMBL3717485) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 9.40E+4 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449864![]() (CHEMBL1491180) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 9.40E+4 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449865![]() (CHEMBL3715535) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.74E+4 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449866![]() (CHEMBL3716352) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.87E+5 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449867![]() (CHEMBL3718612) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 5.93E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449868![]() (CHEMBL3718363) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.33E+4 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449869![]() (CHEMBL3715551) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.34E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449870![]() (CHEMBL3716878) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.74E+4 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449871![]() (CHEMBL3716127) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 5.29E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449872![]() (CHEMBL3717723) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.88E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449873![]() (CHEMBL3716596) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.65E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449874![]() (CHEMBL3717718) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 9.40E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449875![]() (CHEMBL3716813) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 5.29E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449876![]() (CHEMBL3718643) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 8.38E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449877![]() (CHEMBL3716512) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.97E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449878![]() (CHEMBL3719257) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.11E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449879![]() (CHEMBL3715001) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 8.38E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449880![]() (CHEMBL3718178) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 5.93E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449881![]() (CHEMBL3716450) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.32E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449882![]() (CHEMBL3716394) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.88E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449883![]() (CHEMBL3717045) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4.20E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449884![]() (CHEMBL3718895) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.97E+4 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449885![]() (CHEMBL3715266) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 5.93E+4 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Relaxin receptor 1 (Homo sapiens (Human)) | BDBM50449839![]() (CHEMBL3716871) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.65E+3 | n/a | n/a | n/a | n/a |
National Center for Advancing Translational Sciences Curated by ChEMBL | Assay Description Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay | Eur J Med Chem 156: 79-92 (2018) Article DOI: 10.1016/j.ejmech.2018.06.008 BindingDB Entry DOI: 10.7270/Q2474DD4 | |||||||||||
More data for this Ligand-Target Pair |