Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465543![]() (CHEMBL4278778) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 251 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465543![]() (CHEMBL4278778) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 251 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465544![]() (CHEMBL4285802) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 316 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465540![]() (CHEMBL4282396) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 398 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465534![]() (CHEMBL4288560) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 398 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465541![]() (CHEMBL4284735) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 501 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465536![]() (CHEMBL4282793) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 501 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465539![]() (CHEMBL4292433) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 501 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465537![]() (CHEMBL4286225) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 631 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465533![]() (CHEMBL4289190) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 631 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465535![]() (CHEMBL4278314) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 631 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465545![]() (CHEMBL4293000) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 794 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465546![]() (CHEMBL4277865) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 794 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465538![]() (CHEMBL4284197) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465548![]() (CHEMBL4286686) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.26E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465547![]() (CHEMBL4292615) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.59E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465542![]() (CHEMBL4281327) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465551![]() (CHEMBL4290684) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.01E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465549![]() (CHEMBL1721265) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 1.26E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465550![]() (CHEMBL4289645) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.51E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF... | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465546![]() (CHEMBL4277865) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 540 | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetry | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465541![]() (CHEMBL4284735) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 410 | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetry | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465536![]() (CHEMBL4282793) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 890 | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetry | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465535![]() (CHEMBL4278314) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 560 | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetry | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465543![]() (CHEMBL4278778) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetry | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465539![]() (CHEMBL4292433) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 320 | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetry | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465537![]() (CHEMBL4286225) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 590 | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetry | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465533![]() (CHEMBL4289190) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 770 | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetry | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465540![]() (CHEMBL4282396) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 310 | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetry | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465545![]() (CHEMBL4293000) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 860 | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetry | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465538![]() (CHEMBL4284197) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 940 | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetry | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50465544![]() (CHEMBL4285802) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 360 | n/a | n/a | n/a | n/a | n/a |
Aix-Marseille University Curated by ChEMBL | Assay Description Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetry | J Med Chem 61: 5719-5732 (2018) Article DOI: 10.1021/acs.jmedchem.8b00653 BindingDB Entry DOI: 10.7270/Q2Q52S95 | |||||||||||
More data for this Ligand-Target Pair |