Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM69602![]() (2,3-dihydro-1,4-benzodioxin-3-ylmethyl-[2-(2,6-dim...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 0.427 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1A adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM69602![]() (2,3-dihydro-1,4-benzodioxin-3-ylmethyl-[2-(2,6-dim...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 0.513 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1D adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Homo sapiens (Human)) | BDBM50472355![]() (CHEMBL135974) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 0.832 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from human 5-hydroxytryptamine 1A receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Homo sapiens (Human)) | BDBM50026917![]() (8-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-8-a...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 0.933 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from human 5-hydroxytryptamine 1A receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50026917![]() (8-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-8-a...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1D adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Homo sapiens (Human)) | BDBM69602![]() (2,3-dihydro-1,4-benzodioxin-3-ylmethyl-[2-(2,6-dim...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 2.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from human 5-hydroxytryptamine 1A receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Homo sapiens (Human)) | BDBM21393![]() (7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 3.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from human 5-hydroxytryptamine 1A receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Homo sapiens (Human)) | BDBM50472358![]() (CHEMBL132378) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from human 5-hydroxytryptamine 1A receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Homo sapiens (Human)) | BDBM50472353![]() (CHEMBL135973) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 5.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from human 5-hydroxytryptamine 1A receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50472353![]() (CHEMBL135973) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Ability to displace [3H]prazosin from human cloned Alpha-1D adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM69602![]() (2,3-dihydro-1,4-benzodioxin-3-ylmethyl-[2-(2,6-dim...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1B adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor (RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM69602![]() (2,3-dihydro-1,4-benzodioxin-3-ylmethyl-[2-(2,6-dim...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 15 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]rauwolscine from rat brain Alpha-2 adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50472354![]() (CHEMBL134428) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1D adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Homo sapiens (Human)) | BDBM50472354![]() (CHEMBL134428) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 22 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from human 5-hydroxytryptamine 1A receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Homo sapiens (Human)) | BDBM50472357![]() (CHEMBL2112711) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from human 5-hydroxytryptamine 1A receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Homo sapiens (Human)) | BDBM50472357![]() (CHEMBL2112711) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 27 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from human 5-hydroxytryptamine 1A receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Homo sapiens (Human)) | BDBM50472356![]() (CHEMBL2112713) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 33.9 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from human 5-hydroxytryptamine 1A receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Homo sapiens (Human)) | BDBM50472356![]() (CHEMBL2112713) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 34 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from human 5-hydroxytryptamine 1A receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50472353![]() (CHEMBL135973) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 36 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1A adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50472353![]() (CHEMBL135973) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 47 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Ability to displace [3H]prazosin from human cloned Alpha-1B adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50026917![]() (8-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-8-a...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 49 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat brain Dopamine receptor D2 | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50026917![]() (8-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-8-a...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 69 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1B adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50472354![]() (CHEMBL134428) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 78 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1A adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50472354![]() (CHEMBL134428) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 93 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1B adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM69602![]() (2,3-dihydro-1,4-benzodioxin-3-ylmethyl-[2-(2,6-dim...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 123 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat brain Dopamine receptor D2 | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50472355![]() (CHEMBL135974) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1D adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50026917![]() (8-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-8-a...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 380 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1A adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50472355![]() (CHEMBL135974) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 389 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1A adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serotonin 2 (5-HT2) receptor (RAT-Rattus norvegicus (Rat)-Rattus norvegicus (rat...) | BDBM50026917![]() (8-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-8-a...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 490 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]ketanserin from rat brain 5-hydroxytryptamine 2 receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor (RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50472354![]() (CHEMBL134428) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 537 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]rauwolscine from rat brain Alpha-2 adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor (RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50472355![]() (CHEMBL135974) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 589 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]rauwolscine from rat brain Alpha-2 adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor (RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50472358![]() (CHEMBL132378) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 617 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]rauwolscine from rat brain Alpha-2 adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor (RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM21393![]() (7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 832 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]rauwolscine from rat brain Alpha-2 adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor (RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50472353![]() (CHEMBL135973) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 891 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]rauwolscine from rat brain Alpha-2 adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM50472358![]() (CHEMBL132378) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 933 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1D adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM50472358![]() (CHEMBL132378) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 955 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1A adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Homo sapiens (Human)) | BDBM21393![]() (7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1A adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serotonin 2 (5-HT2) receptor (RAT-Rattus norvegicus (Rat)-Rattus norvegicus (rat...) | BDBM50472353![]() (CHEMBL135973) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]ketanserin from rat brain 5-hydroxytryptamine 2 receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50472358![]() (CHEMBL132378) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1B adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serotonin 2 (5-HT2) receptor (RAT-Rattus norvegicus (Rat)-Rattus norvegicus (rat...) | BDBM50472355![]() (CHEMBL135974) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]ketanserin from rat brain 5-hydroxytryptamine 2 receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serotonin 2 (5-HT2) receptor (RAT-Rattus norvegicus (Rat)-Rattus norvegicus (rat...) | BDBM69602![]() (2,3-dihydro-1,4-benzodioxin-3-ylmethyl-[2-(2,6-dim...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]ketanserin from rat brain 5-hydroxytryptamine 2 receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serotonin 2 (5-HT2) receptor (RAT-Rattus norvegicus (Rat)-Rattus norvegicus (rat...) | BDBM21393![]() (7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]ketanserin from rat brain 5-hydroxytryptamine 2 receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Homo sapiens (Human)) | BDBM21393![]() (7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1D adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM21393![]() (7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat brain Dopamine receptor D2 | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM21393![]() (7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1B adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50472358![]() (CHEMBL132378) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 1.12E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat brain Dopamine receptor D2 | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor (RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50026917![]() (8-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-8-a...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 1.18E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]rauwolscine from rat brain Alpha-2 adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Homo sapiens (Human)) | BDBM50472355![]() (CHEMBL135974) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 1.82E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from human cloned Alpha-1B adrenergic receptor | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50472353![]() (CHEMBL135973) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat brain Dopamine receptor D2 | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50472355![]() (CHEMBL135974) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bologna Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat brain Dopamine receptor D2 | J Med Chem 42: 4214-24 (1999) Article DOI: 10.1021/jm991065j BindingDB Entry DOI: 10.7270/Q2TF012V | |||||||||||
More data for this Ligand-Target Pair |
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