Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50260153 (Apamin | CHEMBL525408 | Octadecapeptide venom) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.00400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Li£ge Curated by ChEMBL | Assay Description Displacement of [125I]apamin from Wistar rat cortical apamin-sensitive site | J Med Chem 49: 7208-14 (2006) Article DOI: 10.1021/jm0607395 BindingDB Entry DOI: 10.7270/Q2S75K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50476033 (CHEMBL215533) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 730 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Li£ge Curated by ChEMBL | Assay Description Displacement of [125I]apamin from Wistar rat cortical apamin-sensitive site | J Med Chem 49: 7208-14 (2006) Article DOI: 10.1021/jm0607395 BindingDB Entry DOI: 10.7270/Q2S75K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50476031 (CHEMBL215029) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 910 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Li£ge Curated by ChEMBL | Assay Description Displacement of [125I]apamin from Wistar rat cortical apamin-sensitive site | J Med Chem 49: 7208-14 (2006) Article DOI: 10.1021/jm0607395 BindingDB Entry DOI: 10.7270/Q2S75K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50199404 (1-(3,4-Dimethoxy-benzyl)-6,7-dimethoxy-2,2-dimethy...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Li£ge Curated by ChEMBL | Assay Description Displacement of [125I]apamin from Wistar rat cortical apamin-sensitive site | J Med Chem 49: 7208-14 (2006) Article DOI: 10.1021/jm0607395 BindingDB Entry DOI: 10.7270/Q2S75K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50476029 (CHEMBL215037) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Li£ge Curated by ChEMBL | Assay Description Displacement of [125I]apamin from Wistar rat cortical apamin-sensitive site | J Med Chem 49: 7208-14 (2006) Article DOI: 10.1021/jm0607395 BindingDB Entry DOI: 10.7270/Q2S75K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50476028 (CHEMBL386836 | N-Methyl-Noscapine) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Li£ge Curated by ChEMBL | Assay Description Displacement of [125I]apamin from Wistar rat cortical apamin-sensitive site | J Med Chem 49: 7208-14 (2006) Article DOI: 10.1021/jm0607395 BindingDB Entry DOI: 10.7270/Q2S75K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50476032 (CHEMBL214787) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 5.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Li£ge Curated by ChEMBL | Assay Description Displacement of [125I]apamin from Wistar rat cortical apamin-sensitive site | J Med Chem 49: 7208-14 (2006) Article DOI: 10.1021/jm0607395 BindingDB Entry DOI: 10.7270/Q2S75K20 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50476030 (CHEMBL215382) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 5.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Li£ge Curated by ChEMBL | Assay Description Displacement of [125I]apamin from Wistar rat cortical apamin-sensitive site | J Med Chem 49: 7208-14 (2006) Article DOI: 10.1021/jm0607395 BindingDB Entry DOI: 10.7270/Q2S75K20 | |||||||||||
More data for this Ligand-Target Pair |