Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cytochrome P450 1A2 (Homo sapiens (Human)) | BDBM50510045 (CHEMBL4587871) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of CYP1A2 (unknown origin) using pro-luciferin substrates in presence of NADPH by firefly luciferase reporter gene based P450-Glo assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 1A2 (Homo sapiens (Human)) | BDBM50510038 (CHEMBL4518161) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of CYP1A2 (unknown origin) using pro-luciferin substrates in presence of NADPH by firefly luciferase reporter gene based P450-Glo assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 1A2 (Homo sapiens (Human)) | BDBM50510048 (CHEMBL4442568) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of CYP1A2 (unknown origin) using pro-luciferin substrates in presence of NADPH by firefly luciferase reporter gene based P450-Glo assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510034 (CHEMBL4593063) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 2D6 (Homo sapiens (Human)) | BDBM50510045 (CHEMBL4587871) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of CYP2D6 (unknown origin) using pro-luciferin substrates in presence of NADPH by firefly luciferase reporter gene based P450-Glo assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510054 (CHEMBL4445209) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510045 (CHEMBL4587871) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510054 (CHEMBL4445209) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.25-stimulated mouse ASIC1a/2a heterodimer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence... | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510044 (CHEMBL4462808) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510049 (CHEMBL4590631) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510035 (CHEMBL4528810) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510038 (CHEMBL4518161) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.09E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.25-stimulated mouse ASIC1a/2a heterodimer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence... | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510035 (CHEMBL4528810) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.13E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.25-stimulated mouse ASIC1a/2a heterodimer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence... | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510056 (CHEMBL4450681) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.17E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510036 (CHEMBL4555958) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.56E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510057 (CHEMBL4538655) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.63E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510043 (CHEMBL4524195) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.68E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510048 (CHEMBL4442568) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510038 (CHEMBL4518161) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.89E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 1/2 (Mus musculus) | BDBM50510034 (CHEMBL4593063) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.25-stimulated mouse ASIC1a/2a heterodimer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence... | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510037 (CHEMBL4463769) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50510038 (CHEMBL4518161) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of human ERG incubated for 4 hrs by fluorescence polarization assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 1 (Mus musculus) | BDBM50510034 (CHEMBL4593063) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 1 (Mus musculus) | BDBM50510035 (CHEMBL4528810) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 1 (Mus musculus) | BDBM50510038 (CHEMBL4518161) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 1 (Mus musculus) | BDBM50510039 (CHEMBL4456021) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 1 (Mus musculus) | BDBM50510040 (CHEMBL4469611) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 1 (Mus musculus) | BDBM50510041 (CHEMBL4476781) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 1 (Mus musculus) | BDBM50510042 (CHEMBL4593172) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 1 (Mus musculus) | BDBM50510043 (CHEMBL4524195) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 1 (Mus musculus) | BDBM50510044 (CHEMBL4462808) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 1 (Mus musculus) | BDBM50510045 (CHEMBL4587871) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 1 (Mus musculus) | BDBM50510046 (CHEMBL4440380) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 1 (Mus musculus) | BDBM50510047 (CHEMBL4517411) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 1 (Mus musculus) | BDBM50510048 (CHEMBL4442568) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 1 (Mus musculus) | BDBM50510037 (CHEMBL4463769) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510040 (CHEMBL4469611) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510041 (CHEMBL4476781) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510042 (CHEMBL4593172) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510050 (CHEMBL4463485) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510047 (CHEMBL4517411) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510051 (CHEMBL4527919) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assay | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510039 (CHEMBL4456021) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.25-stimulated mouse ASIC1a/2a heterodimer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence... | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510049 (CHEMBL4590631) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.25-stimulated mouse ASIC1a/2a heterodimer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence... | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510040 (CHEMBL4469611) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.25-stimulated mouse ASIC1a/2a heterodimer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence... | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510052 (CHEMBL4446500) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.25-stimulated mouse ASIC1a/2a heterodimer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence... | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510053 (CHEMBL4591499) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.25-stimulated mouse ASIC1a/2a heterodimer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence... | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510043 (CHEMBL4524195) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.25-stimulated mouse ASIC1a/2a heterodimer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence... | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510036 (CHEMBL4555958) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.25-stimulated mouse ASIC1a/2a heterodimer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence... | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acid-sensing ion channel 2 (Mus musculus) | BDBM50510046 (CHEMBL4440380) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Promidis Curated by ChEMBL | Assay Description Inhibition of pH 6.25-stimulated mouse ASIC1a/2a heterodimer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence... | ACS Med Chem Lett 10: 627-632 (2019) Article DOI: 10.1021/acsmedchemlett.8b00591 BindingDB Entry DOI: 10.7270/Q2RB77Z0 | |||||||||||
More data for this Ligand-Target Pair |
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