Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525948![]() (CHEMBL4516018) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 910 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525947![]() (CHEMBL4560730) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 280 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525950![]() (CHEMBL4552995) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525951![]() (CHEMBL4447367) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525952![]() (CHEMBL4542977) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 670 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525953![]() (CHEMBL4437589) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | n/a | 60 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525954![]() (CHEMBL4474443) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 200 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525955![]() (CHEMBL4455286) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 870 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525956![]() (CHEMBL4465513) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.22E+4 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525957![]() (CHEMBL4461515) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase MCE PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | n/a | 49 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525958![]() (CHEMBL4591600) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.18E+3 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525959![]() (CHEMBL4454987) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.44E+3 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525960![]() (CHEMBL4440011) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 920 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525942![]() (CHEMBL4465567) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 663 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525943![]() (CHEMBL4449850) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4.70E+3 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525944![]() (CHEMBL4585693) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 740 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525945![]() (CHEMBL4449495) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 125 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525946![]() (CHEMBL4586856) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.06E+3 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel subfamily V member 4 (Homo sapiens (Human)) | BDBM50525949![]() (CHEMBL4436655) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a |
Asahi Kasei Medical Corporation Curated by ChEMBL | Assay Description Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/... | J Med Chem 62: 1468-1483 (2019) Article DOI: 10.1021/acs.jmedchem.8b01615 BindingDB Entry DOI: 10.7270/Q2HD803S | |||||||||||
More data for this Ligand-Target Pair |