Found 35 hits Enz. Inhib. hit(s) with all data for entry = 50011773 Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM11162
((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)Show SMILES N[C@@H](CC(=O)N1CCn2c(C1)nnc2C(F)(F)F)Cc1cc(F)c(F)cc1F |r| Show InChI InChI=1S/C16H15F6N5O/c17-10-6-12(19)11(18)4-8(10)3-9(23)5-14(28)26-1-2-27-13(7-26)24-25-15(27)16(20,21)22/h4,6,9H,1-3,5,7,23H2/t9-/m1/s1 | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
| Purchase
CHEMBL
DrugBank
MCE
PC cid
PC sid
PDB
UniChem
Similars
| DrugBank
PDB
Article
PubMed
| n/a | n/a | 8.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | 
3D Structure (crystal) |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550973
(CHEMBL4784857)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3nc(no3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| Purchase
MCE
PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550969
(CHEMBL4744389)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCC(CC3)c3nc(c[nH]3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 44 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550967
(CHEMBL4762199)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCC(CC3)n3cc(nn3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 47 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550977
(CHEMBL4740282)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3nc(cs3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 59 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550975
(CHEMBL4742337)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3nnc([nH]3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 76 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550976
(CHEMBL4799779)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3cc(C)nn3-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 83 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550970
(CHEMBL4750433)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCC(CC3)c3ncc(o3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550968
(CHEMBL4743350)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCC(CC3)c3nc(cs3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550971
(CHEMBL4783756)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCC(CC3)c3cc(on3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550966
(CHEMBL4761281)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCC(CC3)c3nc(no3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550972
(CHEMBL4796411)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCC(CC3)c3nnnn3-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 270 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550983
(CHEMBL4749117)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3ncc(F)cn3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 350 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550974
(CHEMBL4795875)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3nc(ns3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 360 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550982
(CHEMBL4764779)Show SMILES COc1cnc(nc1)N1CCN(CCCn2c(=O)n(C)c3nc(N4CCC[C@@H](N)C4)n(CC#CC)c3c2=O)CC1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 430 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550981
(CHEMBL4776485)Show SMILES CCCc1cnc(nc1)N1CCN(CCCn2c(=O)n(C)c3nc(N4CCC[C@@H](N)C4)n(CC#CC)c3c2=O)CC1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 590 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550980
(CHEMBL4745258)Show SMILES CCc1cnc(nc1)N1CCN(CCCn2c(=O)n(C)c3nc(N4CCC[C@@H](N)C4)n(CC#CC)c3c2=O)CC1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 610 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550979
(CHEMBL4785060)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3ncc(C)cn3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 660 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550978
(CHEMBL4782382)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3noc(n3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 680 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Dipeptidyl peptidase 4
(Homo sapiens (Human)) | BDBM50550984
(CHEMBL4751384)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3ncc(cn3)C(F)(F)F)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 740 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hr |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Potassium voltage-gated channel subfamily H member 2
(Homo sapiens (Human)) | BDBM50550973
(CHEMBL4784857)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3nc(no3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| Purchase
MCE
PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 4.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of human ERG expressed in CHO cells by manual patch clamp assay |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Glucose-dependent insulinotropic receptor
(Homo sapiens (Human)) | BDBM50244791
((2-Fluoro-4-methanesulfonyl-phenyl)-{6-[4-(3-isopr...)Show SMILES CC(C)c1nc([o+][n-]1)C1CCN(CC1)c1ncnc(Nc2ccc(cc2F)S(C)(=O)=O)c1[N+]([O-])=O Show InChI InChI=1S/C21H24FN7O5S/c1-12(2)18-26-21(34-27-18)13-6-8-28(9-7-13)20-17(29(30)31)19(23-11-24-20)25-16-5-4-14(10-15(16)22)35(3,32)33/h4-5,10-13H,6-9H2,1-3H3,(H,23,24,25) | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| Purchase
CHEMBL
MCE
PC cid
PC sid
UniChem
Patents
Similars
| Article
PubMed
| n/a | n/a | n/a | n/a | 640 | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assay |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Glucose-dependent insulinotropic receptor
(Homo sapiens (Human)) | BDBM50550979
(CHEMBL4785060)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3ncc(C)cn3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | n/a | n/a | 2.56E+3 | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assay |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Glucose-dependent insulinotropic receptor
(Homo sapiens (Human)) | BDBM50550980
(CHEMBL4745258)Show SMILES CCc1cnc(nc1)N1CCN(CCCn2c(=O)n(C)c3nc(N4CCC[C@@H](N)C4)n(CC#CC)c3c2=O)CC1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | n/a | n/a | 3.99E+3 | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assay |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Glucose-dependent insulinotropic receptor
(Homo sapiens (Human)) | BDBM50550981
(CHEMBL4776485)Show SMILES CCCc1cnc(nc1)N1CCN(CCCn2c(=O)n(C)c3nc(N4CCC[C@@H](N)C4)n(CC#CC)c3c2=O)CC1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | n/a | n/a | 1.85E+3 | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assay |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Glucose-dependent insulinotropic receptor
(Homo sapiens (Human)) | BDBM50550982
(CHEMBL4764779)Show SMILES COc1cnc(nc1)N1CCN(CCCn2c(=O)n(C)c3nc(N4CCC[C@@H](N)C4)n(CC#CC)c3c2=O)CC1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | n/a | n/a | 2.26E+3 | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assay |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Glucose-dependent insulinotropic receptor
(Homo sapiens (Human)) | BDBM50550983
(CHEMBL4749117)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3ncc(F)cn3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | n/a | n/a | 1.41E+3 | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assay |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Glucose-dependent insulinotropic receptor
(Homo sapiens (Human)) | BDBM50550984
(CHEMBL4751384)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3ncc(cn3)C(F)(F)F)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | n/a | n/a | 4.02E+3 | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assay |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Glucose-dependent insulinotropic receptor
(Homo sapiens (Human)) | BDBM50550978
(CHEMBL4782382)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3noc(n3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | n/a | n/a | 1.45E+3 | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assay |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Glucose-dependent insulinotropic receptor
(Homo sapiens (Human)) | BDBM50550977
(CHEMBL4740282)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3nc(cs3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | n/a | n/a | 650 | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assay |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Glucose-dependent insulinotropic receptor
(Homo sapiens (Human)) | BDBM50550973
(CHEMBL4784857)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3nc(no3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| Purchase
MCE
PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assay |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Glucose-dependent insulinotropic receptor
(Homo sapiens (Human)) | BDBM50550970
(CHEMBL4750433)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCC(CC3)c3ncc(o3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | n/a | n/a | 830 | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assay |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Glucose-dependent insulinotropic receptor
(Homo sapiens (Human)) | BDBM50550969
(CHEMBL4744389)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCC(CC3)c3nc(c[nH]3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | n/a | n/a | 600 | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assay |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Glucose-dependent insulinotropic receptor
(Homo sapiens (Human)) | BDBM50550968
(CHEMBL4743350)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCC(CC3)c3nc(cs3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | n/a | n/a | 3.13E+3 | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assay |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
Glucose-dependent insulinotropic receptor
(Homo sapiens (Human)) | BDBM50550974
(CHEMBL4795875)Show SMILES CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3nc(ns3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1 |r| | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | n/a | n/a | 1.93E+3 | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assay |
Citation and Details
Article DOI: 10.1016/j.ejmech.2019.112017
BindingDB Entry DOI: 10.7270/Q2V98CP1 |
More data for this
Ligand-Target Pair | |
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