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Compile Data Set for Download or QSAR

Found 41 hits Enz. Inhib. hit(s) with all data for entry = 50011817   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551405
PNG
(CHEMBL4784488)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccc(F)c(Cl)c1)c1ccc(C)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
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PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 520n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551445
PNG
(CHEMBL4782169)
Show SMILES [H][C@@]12[C@H](O)[C@H](OC(C)=O)[C@@]3(C)C[C@](C)(CC(=O)[C@]3(O)C1[C@@H](O)CCC2(C)C)C=C |r|
PDB

UniProtKB/SwissProt

antibodypedia
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UniChem
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n/an/an/an/a 1.46E+4n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551407
PNG
(CHEMBL4786932)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccc(C)cc1F)c1ccc(C)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 770n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551408
PNG
(CHEMBL4761430)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccc(C)cc1OC)c1cccc(C)c1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
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UniChem
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PubMed
n/an/an/an/a 5.96E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551409
PNG
(CHEMBL4789237)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccc(C)cc1)c1ccc(CC)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 670n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551410
PNG
(CHEMBL4760850)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccc(F)cc1)c1ccc(cc1)C(C)C |r|
PDB

UniProtKB/SwissProt

antibodypedia
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UniChem
Article
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n/an/an/an/a 1.30E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551411
PNG
(CHEMBL4759872)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccc(OCC)cc1)c1ccc(F)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
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UniChem
Article
PubMed
n/an/an/an/a 3.93E+4n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551412
PNG
(CHEMBL4764988)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccc(CC)cc1)c1ccc(Cl)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 430n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551413
PNG
(CHEMBL4742351)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1cccc(F)c1)c1ccc(Cl)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
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PC sid
UniChem
Article
PubMed
n/an/an/an/a 3.53E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551414
PNG
(CHEMBL4779970)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccc(F)cc1)c1ccc(Cl)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 530n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551415
PNG
(CHEMBL4744648)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1cc(C)cc(C)c1)c1ccc(Cl)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 310n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551416
PNG
(CHEMBL4798759)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccc(C)cc1)c1cccc(Cl)c1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 5.05E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551417
PNG
(CHEMBL4787822)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccc(C)cc1)c1ccc(OCC)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
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PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 2.48E+4n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551418
PNG
(CHEMBL4760156)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccc(C)cc1)c1cccc(OC)c1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 1.60E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551419
PNG
(CHEMBL4751807)
Show SMILES [H][C@]12[C@@H](CCC)OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccccc1Cl |r|
PDB

UniProtKB/SwissProt

antibodypedia
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PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 4.29E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551420
PNG
(CHEMBL4745662)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C)C2=O)c1ccc(C)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
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PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 3.08E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551421
PNG
(CHEMBL4747654)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C(C)C)C2=O)c1ccc(C)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
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UniChem
Article
PubMed
n/an/an/an/a 7.34E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551422
PNG
(CHEMBL4761233)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C1CC1)C2=O)c1ccc(C)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 3.37E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551423
PNG
(CHEMBL4795137)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C1CCCC1)C2=O)c1ccc(C)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 3.44E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551424
PNG
(CHEMBL4754971)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C1CCCCC1)C2=O)c1ccc(C)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 1.29E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551425
PNG
(CHEMBL4761309)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccc(C)cc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccccc1Cl)c1ccc(C)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 300n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551426
PNG
(CHEMBL4751732)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccc(Br)cc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccccc1Cl)c1ccc(C)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
Purchase

MCE
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 90n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551427
PNG
(CHEMBL4777571)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccc(Cl)cc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccccc1Cl)c1ccc(C)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 236n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551428
PNG
(CHEMBL4744718)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccc(F)cc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccccc1Cl)c1ccc(C)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
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PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 692n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551429
PNG
(CHEMBL4760543)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4cccc(C)c4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccccc1Cl)c1ccc(C)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 1.08E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551430
PNG
(CHEMBL4781262)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4cccc(Br)c4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccccc1Cl)c1ccc(C)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 1.16E+4n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551431
PNG
(CHEMBL4762531)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4cccc(Cl)c4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccccc1Cl)c1ccc(C)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 301n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551432
PNG
(CHEMBL4758446)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4cccc(F)c4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccccc1Cl)c1ccc(C)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 345n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551433
PNG
(CHEMBL4800693)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccc(Cl)cc1)c1ccccc1 |r|
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n/an/an/an/a 2.06E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551434
PNG
(CHEMBL4799136)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1cc(Cl)ccc1C)c1ccccc1 |r|
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n/an/an/an/a 3.12E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551435
PNG
(CHEMBL4794886)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1cccc(Cl)c1)c1ccccc1 |r|
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n/an/an/an/a 8.10E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551436
PNG
(CHEMBL4754188)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1cc(OC)ccc1OC)c1ccc(C)cc1 |r|
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n/an/an/an/a 1.20E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551437
PNG
(CHEMBL4745564)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccc(OCC)cc1)c1ccccc1 |r|
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n/an/an/an/a 3.23E+4n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551438
PNG
(CHEMBL4750740)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccccc1Cl)c1ccc(C)cc1 |r|
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n/an/an/an/a 170n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551439
PNG
(CHEMBL4763027)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccccc1Cl)c1cccc(C)c1 |r|
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n/an/an/an/a 6.81E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551440
PNG
(CHEMBL4751176)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccc(F)cc1)c1ccc(C)cc1 |r|
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n/an/an/an/a 1.64E+3n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551441
PNG
(CHEMBL4745593)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccc(C)c(Cl)c1)c1ccc(C)cc1 |r|
PDB

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n/an/an/an/a 750n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551442
PNG
(CHEMBL4800461)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccc(OC)cc1)c1ccc(C)cc1 |r|
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n/an/an/an/a 1.71E+4n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551443
PNG
(CHEMBL4743444)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccc(OCC)cc1)c1ccc(C)cc1 |r|
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n/an/an/an/a 1.08E+4n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551444
PNG
(CHEMBL4763908)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1cccc(OC)c1)c1ccc(C)cc1 |r|
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n/an/an/an/a 960n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair
Adenylate cyclase type 2


(Homo sapiens (Human))
BDBM50551406
PNG
(CHEMBL4740707)
Show SMILES [H][C@]12[C@H](OC3(C(=O)c4ccccc4C3=O)[C@@]1([H])C(=O)N(C2=O)c1ccc(C)c(C)c1)c1ccc(C)cc1 |r|
PDB

UniProtKB/SwissProt

antibodypedia
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n/an/an/an/a 210n/an/an/an/a


TBA

Assay Description
Agonist activity at recombinant human AC2 expressed in HEK293 cells assessed as increase in cAMP level measured after 30 mins by LANCE Ultra cAMP Det...


Citation and Details

Article DOI: 10.1016/j.ejmech.2020.112115
BindingDB Entry DOI: 10.7270/Q27D2ZR4
More data for this
Ligand-Target Pair