Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111082![]() (9-Chloro-2-phenyl-3,4,5,6-tetrahydro-1,3-diaza-ben...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111079![]() (9-Methyl-2-pyridin-3-yl-3,4,5,6-tetrahydro-1,3-dia...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111085![]() (2-Phenyl-3,4,5,6-tetrahydro-1,3-diaza-benzo[e]azul...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111083![]() (9-Methoxy-2-pyridin-3-yl-3,4,5,6-tetrahydro-1,3-di...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 6.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111089![]() (9-Methyl-2-pyridin-4-yl-3,4,5,6-tetrahydro-1,3-dia...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 6.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111092![]() (9-Fluoro-2-pyridin-3-yl-3,4,5,6-tetrahydro-1,3-dia...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 6.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111094![]() (2-Pyridin-3-yl-3,4,5,6-tetrahydro-1,3-diaza-benzo[...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 7.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111095![]() (9-Methoxy-2-pyridin-4-yl-3,4,5,6-tetrahydro-1,3-di...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111080![]() (9-Fluoro-2-pyridin-4-yl-3,4,5,6-tetrahydro-1,3-dia...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111081![]() (2-Pyridin-4-yl-3,4,5,6-tetrahydro-1,3-diaza-benzo[...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111096![]() (9-Methoxy-2-phenyl-3,4,5,6-tetrahydro-1,3-diaza-be...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111078![]() (9-Methyl-2-pyridin-2-yl-3,4,5,6-tetrahydro-1,3-dia...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 32 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111088![]() (9-Fluoro-2-pyridin-2-yl-3,4,5,6-tetrahydro-1,3-dia...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 46 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111090![]() (8-Methoxy-2-phenyl-4,5-dihydro-3H-naphtho[1,2-d]im...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 52 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111087![]() (9-Methoxy-2-pyridin-2-yl-3,4,5,6-tetrahydro-1,3-di...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111091![]() (2-Pyridin-2-yl-3,4,5,6-tetrahydro-1,3-diaza-benzo[...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111086![]() (3-(5-Methyl-2-phenyl-1H-imidazol-4-yl)-pyridine | ...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 427 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111093![]() (2-(1H-Imidazol-4-yl)-3,4,5,6-tetrahydro-1,3-diaza-...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 570 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50111084![]() (2-Phenyl-4,5-dihydro-3H-6-oxa-1,3-diaza-benzo[e]az...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 6.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co., Ltd. Curated by ChEMBL | Assay Description Concentration that inhibited 50% of binding of 125 I -PYY ligand to human Neuropeptide Y receptor type 5 | Bioorg Med Chem Lett 12: 1009-11 (2002) BindingDB Entry DOI: 10.7270/Q2J102G1 | |||||||||||
More data for this Ligand-Target Pair |