Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552240 (CHEMBL4780197) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 120 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Mixed type inhibition of porcine pancreatic lipase using 4MUO as substrate by Lineweaver-Burk plot analysis | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552242 (CHEMBL365190) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.70 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552240 (CHEMBL4780197) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 330 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552238 (CHEMBL4788400) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 580 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552241 (CHEMBL4797179) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 680 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552236 (CHEMBL4782276) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 830 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552233 (CHEMBL4748399) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.69E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552234 (CHEMBL4757866) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.09E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552237 (CHEMBL4744746) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.52E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552229 (CHEMBL4752404) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.54E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552231 (CHEMBL4740149) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.32E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552232 (CHEMBL4776624) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552212 (CHEMBL4761197) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.94E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552230 (CHEMBL4745825) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.61E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552214 (CHEMBL4747287) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.04E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552215 (CHEMBL4751728) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.24E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552217 (CHEMBL4778007) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.48E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552222 (CHEMBL4080900) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.48E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552213 (CHEMBL4160838) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.49E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552218 (CHEMBL4780689) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.07E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552216 (CHEMBL4765140) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.48E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552235 (CHEMBL4750178) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.51E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552221 (CHEMBL4098933) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.89E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552226 (CHEMBL4086755) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.27E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552220 (CHEMBL4742119) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552228 (CHEMBL4756815) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.72E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552225 (CHEMBL4779689) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.54E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552223 (CHEMBL4091194) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.56E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552239 (CHEMBL4747550) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.41E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM29143 (CHEMBL7976 | Chalcone 1 | Chalcone, 13 | cid_63776...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.44E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552224 (CHEMBL4785507) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552227 (CHEMBL4078900) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Pancreatic triacylglycerol lipase (Sus scrofa (Pig)) | BDBM50552219 (CHEMBL4170979) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine pancreatic lipase preincubated for 10 mins followed by 4-MUO addition and measured at 60 sec interval for 40 mins by multi plat... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115853 BindingDB Entry DOI: 10.7270/Q2DV1PJS | |||||||||||
More data for this Ligand-Target Pair |