Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Activin receptor type-1 (Homo sapiens (Human)) | BDBM50557476 (CHEMBL4748071) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Louisiana at Monroe Curated by ChEMBL | Assay Description Inhibition of human ALK2 R206H mutant using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot assay | Bioorg Med Chem Lett 12: 2743-7 (2002) Article DOI: 10.1016/j.bmcl.2021.127858 BindingDB Entry DOI: 10.7270/Q25M69C9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Activin receptor type-1 (Homo sapiens (Human)) | BDBM50557474 (CHEMBL4744674) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Louisiana at Monroe Curated by ChEMBL | Assay Description Inhibition of human ALK2 R206H mutant using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot assay | Bioorg Med Chem Lett 12: 2743-7 (2002) Article DOI: 10.1016/j.bmcl.2021.127858 BindingDB Entry DOI: 10.7270/Q25M69C9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Activin receptor type-1 (Homo sapiens (Human)) | BDBM50557481 (CHEMBL4749744) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Louisiana at Monroe Curated by ChEMBL | Assay Description Inhibition of human ALK2 R206H mutant using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot assay | Bioorg Med Chem Lett 12: 2743-7 (2002) Article DOI: 10.1016/j.bmcl.2021.127858 BindingDB Entry DOI: 10.7270/Q25M69C9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Activin receptor type-1 (Homo sapiens (Human)) | BDBM50557475 (CHEMBL4776838) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Louisiana at Monroe Curated by ChEMBL | Assay Description Inhibition of human ALK2 R206H mutant using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot assay | Bioorg Med Chem Lett 12: 2743-7 (2002) Article DOI: 10.1016/j.bmcl.2021.127858 BindingDB Entry DOI: 10.7270/Q25M69C9 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Activin receptor type-1 (Homo sapiens (Human)) | BDBM50557480 (CHEMBL4797111) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 29 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Louisiana at Monroe Curated by ChEMBL | Assay Description Inhibition of human ALK2 R206H mutant using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot assay | Bioorg Med Chem Lett 12: 2743-7 (2002) Article DOI: 10.1016/j.bmcl.2021.127858 BindingDB Entry DOI: 10.7270/Q25M69C9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Activin receptor type-1 (Homo sapiens (Human)) | BDBM50557473 (CHEMBL4749510) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 66 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Louisiana at Monroe Curated by ChEMBL | Assay Description Inhibition of human ALK2 R206H mutant using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot assay | Bioorg Med Chem Lett 12: 2743-7 (2002) Article DOI: 10.1016/j.bmcl.2021.127858 BindingDB Entry DOI: 10.7270/Q25M69C9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Activin receptor type-1 (Homo sapiens (Human)) | BDBM50557472 (CHEMBL4747414) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 167 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Louisiana at Monroe Curated by ChEMBL | Assay Description Inhibition of human ALK2 R206H mutant using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot assay | Bioorg Med Chem Lett 12: 2743-7 (2002) Article DOI: 10.1016/j.bmcl.2021.127858 BindingDB Entry DOI: 10.7270/Q25M69C9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Activin receptor type-1 (Homo sapiens (Human)) | BDBM50557477 (CHEMBL4760836) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 276 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Louisiana at Monroe Curated by ChEMBL | Assay Description Inhibition of human ALK2 R206H mutant using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot assay | Bioorg Med Chem Lett 12: 2743-7 (2002) Article DOI: 10.1016/j.bmcl.2021.127858 BindingDB Entry DOI: 10.7270/Q25M69C9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Activin receptor type-1 (Homo sapiens (Human)) | BDBM50557478 (CHEMBL4793870) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 665 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Louisiana at Monroe Curated by ChEMBL | Assay Description Inhibition of human ALK2 R206H mutant using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot assay | Bioorg Med Chem Lett 12: 2743-7 (2002) Article DOI: 10.1016/j.bmcl.2021.127858 BindingDB Entry DOI: 10.7270/Q25M69C9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Activin receptor type-1 (Homo sapiens (Human)) | BDBM50557471 (CHEMBL4798765) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | 684 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Louisiana at Monroe Curated by ChEMBL | Assay Description Inhibition of human ALK2 R206H mutant using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot assay | Bioorg Med Chem Lett 12: 2743-7 (2002) Article DOI: 10.1016/j.bmcl.2021.127858 BindingDB Entry DOI: 10.7270/Q25M69C9 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Activin receptor type-1 (Homo sapiens (Human)) | BDBM50557479 (CHEMBL4799263) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.89E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Louisiana at Monroe Curated by ChEMBL | Assay Description Inhibition of human ALK2 R206H mutant using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot assay | Bioorg Med Chem Lett 12: 2743-7 (2002) Article DOI: 10.1016/j.bmcl.2021.127858 BindingDB Entry DOI: 10.7270/Q25M69C9 | |||||||||||
More data for this Ligand-Target Pair |