Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Protein ADM2 (Homo sapiens (Human)) | BDBM50570409![]() (CHEMBL4857810) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.631 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570408![]() (CHEMBL4873687) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.631 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570410![]() (CHEMBL4851152) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570410![]() (CHEMBL4851152) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570413![]() (CHEMBL4850259) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570411![]() (CHEMBL4877585) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.60 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570411![]() (CHEMBL4877585) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570401![]() (CHEMBL4879142) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570404![]() (CHEMBL4850583) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570396![]() (CHEMBL4871934) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570409![]() (CHEMBL4857810) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570395![]() (CHEMBL4866915) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570397![]() (CHEMBL4852669) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570398![]() (CHEMBL4861626) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570413![]() (CHEMBL4850259) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570396![]() (CHEMBL4871934) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570397![]() (CHEMBL4852669) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570403![]() (CHEMBL4874651) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570394![]() (CHEMBL4866548) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570406![]() (CHEMBL4862324) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570401![]() (CHEMBL4879142) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 32 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570400![]() (CHEMBL4876643) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570400![]() (CHEMBL4876643) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 79 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570393![]() (CHEMBL4878394) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570390![]() (CHEMBL4851106) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570402![]() (CHEMBL4856402) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570392![]() (CHEMBL4870543) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570408![]() (CHEMBL4873687) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570402![]() (CHEMBL4856402) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 126 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570404![]() (CHEMBL4850583) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 126 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570398![]() (CHEMBL4861626) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 126 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570388![]() (CHEMBL4858139) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570412![]() (CHEMBL4853766) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570394![]() (CHEMBL4866548) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 316 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570395![]() (CHEMBL4866915) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 316 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570405![]() (CHEMBL4874859) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 398 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570406![]() (CHEMBL4862324) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 501 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570407![]() (CHEMBL4865654) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 501 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570412![]() (CHEMBL4853766) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 794 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570399![]() (CHEMBL4846989) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 794 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570405![]() (CHEMBL4874859) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570390![]() (CHEMBL4851106) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570393![]() (CHEMBL4878394) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570403![]() (CHEMBL4874651) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.26E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570386![]() (CHEMBL4864804) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.26E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570407![]() (CHEMBL4865654) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570399![]() (CHEMBL4846989) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.16E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calcitonin gene-related peptide 2 (Homo sapiens) | BDBM50570391![]() (CHEMBL4876213) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.16E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human CGRP-2 (8 to 37 residues) expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preinc... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570392![]() (CHEMBL4870543) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.94E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein ADM2 (Homo sapiens (Human)) | BDBM50570391![]() (CHEMBL4876213) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02191 BindingDB Entry DOI: 10.7270/Q2474FM7 | |||||||||||
More data for this Ligand-Target Pair |
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