BindingDB PrimarySearch

Found 2 hits Enz. Inhib. hit(s) with all data for entry = 50040280
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT)	BDBM50316373 (Argiotoxin-636 \| CHEMBL1098240) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	74	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of rat GluN1/2A expressed in xenopus laevis oocytes assessed as inhibition of glycine-evoked current at membrane potential of -60 mV by vo...				J Nat Prod 74: 483-6 (2011) Article DOI: 10.1021/np100746w BindingDB Entry DOI: 10.7270/Q2KK9CWC
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair
Glutamate receptor 1 (Rattus norvegicus (Rat))	BDBM50316373 (Argiotoxin-636 \| CHEMBL1098240) Show SMILES Show InChI	PDB UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	77	n/a	n/a	n/a	n/a	n/a	n/a
University of Copenhagen Curated by ChEMBL					Assay Description Inhibition of rat GluA1 expressed in xenopus laevis oocytes assessed as inhibition of glutamate-evoked current at membrane potential of -60 mV by vol...				J Nat Prod 74: 483-6 (2011) Article DOI: 10.1021/np100746w BindingDB Entry DOI: 10.7270/Q2KK9CWC
University of Copenhagen Curated by ChEMBL					More data for this Ligand-Target Pair