Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM21147![]() ((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.320 | n/a | n/a | n/a | n/a | n/a | n/a |
Glaxo Wellcome Curated by ChEMBL | Assay Description Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type B receptor stably expressed in CHO-K1 cells | J Med Chem 39: 562-9 (1996) Article DOI: 10.1021/jm950626d BindingDB Entry DOI: 10.7270/Q22R3SZ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM21147![]() ((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.630 | n/a | n/a | n/a | n/a | n/a | n/a |
Glaxo Wellcome Curated by ChEMBL | Assay Description Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type A receptor stably expressed in CHO-K1 cells | J Med Chem 39: 562-9 (1996) Article DOI: 10.1021/jm950626d BindingDB Entry DOI: 10.7270/Q22R3SZ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50422155![]() (CHEMBL443825) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Glaxo Wellcome Curated by ChEMBL | Assay Description Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type B receptor expressed in CHO-K1 cells | J Med Chem 39: 562-9 (1996) Article DOI: 10.1021/jm950626d BindingDB Entry DOI: 10.7270/Q22R3SZ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50072427![]() (1-(1-(2-(isopropyl(phenyl)amino)-2-oxoethyl)-2,4-d...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
Glaxo Wellcome Curated by ChEMBL | Assay Description Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type B receptor expressed in CHO-K1 cells | J Med Chem 39: 562-9 (1996) Article DOI: 10.1021/jm950626d BindingDB Entry DOI: 10.7270/Q22R3SZ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50422157![]() (CHEMBL345786) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 32 | n/a | n/a | n/a | n/a | n/a | n/a |
Glaxo Wellcome Curated by ChEMBL | Assay Description Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type B receptor expressed in CHO-K1 cells | J Med Chem 39: 562-9 (1996) Article DOI: 10.1021/jm950626d BindingDB Entry DOI: 10.7270/Q22R3SZ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50422156![]() (CHEMBL346179) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Glaxo Wellcome Curated by ChEMBL | Assay Description Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type B receptor expressed in CHO-K1 cells | J Med Chem 39: 562-9 (1996) Article DOI: 10.1021/jm950626d BindingDB Entry DOI: 10.7270/Q22R3SZ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50422155![]() (CHEMBL443825) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Glaxo Wellcome Curated by ChEMBL | Assay Description Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type A receptor stably expressed in CHO-K1 cells | J Med Chem 39: 562-9 (1996) Article DOI: 10.1021/jm950626d BindingDB Entry DOI: 10.7270/Q22R3SZ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50072427![]() (1-(1-(2-(isopropyl(phenyl)amino)-2-oxoethyl)-2,4-d...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
Glaxo Wellcome Curated by ChEMBL | Assay Description Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type A receptor stably expressed in CHO-K1 cells | J Med Chem 39: 562-9 (1996) Article DOI: 10.1021/jm950626d BindingDB Entry DOI: 10.7270/Q22R3SZ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50072425![]() (2-[2,4-Dioxo-5-phenyl-3-(3-phenyl-ureido)-2,3,4,5-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
Glaxo Wellcome Curated by ChEMBL | Assay Description Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type B receptor expressed in CHO-K1 cells | J Med Chem 39: 562-9 (1996) Article DOI: 10.1021/jm950626d BindingDB Entry DOI: 10.7270/Q22R3SZ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50422153![]() (CHEMBL345869) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 63 | n/a | n/a | n/a | n/a | n/a | n/a |
Glaxo Wellcome Curated by ChEMBL | Assay Description Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type A receptor stably expressed in CHO-K1 cells | J Med Chem 39: 562-9 (1996) Article DOI: 10.1021/jm950626d BindingDB Entry DOI: 10.7270/Q22R3SZ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50072425![]() (2-[2,4-Dioxo-5-phenyl-3-(3-phenyl-ureido)-2,3,4,5-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 79 | n/a | n/a | n/a | n/a | n/a | n/a |
Glaxo Wellcome Curated by ChEMBL | Assay Description Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type A receptor stably expressed in CHO-K1 cells | J Med Chem 39: 562-9 (1996) Article DOI: 10.1021/jm950626d BindingDB Entry DOI: 10.7270/Q22R3SZ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50422157![]() (CHEMBL345786) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
Glaxo Wellcome Curated by ChEMBL | Assay Description Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type A receptor stably expressed in CHO-K1 cells | J Med Chem 39: 562-9 (1996) Article DOI: 10.1021/jm950626d BindingDB Entry DOI: 10.7270/Q22R3SZ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50422154![]() (CHEMBL154615) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 158 | n/a | n/a | n/a | n/a | n/a | n/a |
Glaxo Wellcome Curated by ChEMBL | Assay Description Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type B receptor expressed in CHO-K1 cells | J Med Chem 39: 562-9 (1996) Article DOI: 10.1021/jm950626d BindingDB Entry DOI: 10.7270/Q22R3SZ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50422153![]() (CHEMBL345869) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 251 | n/a | n/a | n/a | n/a | n/a | n/a |
Glaxo Wellcome Curated by ChEMBL | Assay Description Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type B receptor expressed in CHO-K1 cells | J Med Chem 39: 562-9 (1996) Article DOI: 10.1021/jm950626d BindingDB Entry DOI: 10.7270/Q22R3SZ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50422154![]() (CHEMBL154615) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Glaxo Wellcome Curated by ChEMBL | Assay Description Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type A receptor stably expressed in CHO-K1 cells | J Med Chem 39: 562-9 (1996) Article DOI: 10.1021/jm950626d BindingDB Entry DOI: 10.7270/Q22R3SZ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50422156![]() (CHEMBL346179) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.51E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Glaxo Wellcome Curated by ChEMBL | Assay Description Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type A receptor stably expressed in CHO-K1 cells | J Med Chem 39: 562-9 (1996) Article DOI: 10.1021/jm950626d BindingDB Entry DOI: 10.7270/Q22R3SZ1 | |||||||||||
More data for this Ligand-Target Pair |