Found 64 hits Enz. Inhib. hit(s) with all data for entry = 50042499 Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50426906
(CHEMBL2323692)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)CO)cc1 |r| Show InChI InChI=1S/C27H41N3O8/c1-15(2)21-18(25(30-29-21)38-26-24(36)23(35)22(34)19(13-31)37-26)12-17-10-8-16(9-11-17)6-5-7-20(33)28-27(3,4)14-32/h8-11,15,19,22-24,26,31-32,34-36H,5-7,12-14H2,1-4H3,(H,28,33)(H,29,30)/t19-,22-,23+,24-,26+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet 
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426894
(CHEMBL2323684)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)N2CCN(C)CC2)cc1 |r| Show InChI InChI=1S/C32H49N5O8/c1-19(2)25-22(29(35-34-25)45-30-28(42)27(41)26(40)23(18-38)44-30)17-21-11-9-20(10-12-21)7-6-8-24(39)33-32(3,4)31(43)37-15-13-36(5)14-16-37/h9-12,19,23,26-28,30,38,40-42H,6-8,13-18H2,1-5H3,(H,33,39)(H,34,35)/t23-,26-,27+,28-,30+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426887
(CHEMBL2323695)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)N2CCNCC2)cc1C |r| Show InChI InChI=1S/C32H49N5O8/c1-18(2)25-22(29(36-35-25)45-30-28(42)27(41)26(40)23(17-38)44-30)16-21-10-9-20(15-19(21)3)7-6-8-24(39)34-32(4,5)31(43)37-13-11-33-12-14-37/h9-10,15,18,23,26-28,30,33,38,40-42H,6-8,11-14,16-17H2,1-5H3,(H,34,39)(H,35,36)/t23-,26-,27+,28-,30+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426906
(CHEMBL2323692)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)CO)cc1 |r| Show InChI InChI=1S/C27H41N3O8/c1-15(2)21-18(25(30-29-21)38-26-24(36)23(35)22(34)19(13-31)37-26)12-17-10-8-16(9-11-17)6-5-7-20(33)28-27(3,4)14-32/h8-11,15,19,22-24,26,31-32,34-36H,5-7,12-14H2,1-4H3,(H,28,33)(H,29,30)/t19-,22-,23+,24-,26+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426895
(CHEMBL2323683)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)N2CCNCC2)cc1 |r| Show InChI InChI=1S/C31H47N5O8/c1-18(2)24-21(28(35-34-24)44-29-27(41)26(40)25(39)22(17-37)43-29)16-20-10-8-19(9-11-20)6-5-7-23(38)33-31(3,4)30(42)36-14-12-32-13-15-36/h8-11,18,22,25-27,29,32,37,39-41H,5-7,12-17H2,1-4H3,(H,33,38)(H,34,35)/t22-,25-,26+,27-,29+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50426894
(CHEMBL2323684)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)N2CCN(C)CC2)cc1 |r| Show InChI InChI=1S/C32H49N5O8/c1-19(2)25-22(29(35-34-25)45-30-28(42)27(41)26(40)23(18-38)44-30)17-21-11-9-20(10-12-21)7-6-8-24(39)33-32(3,4)31(43)37-15-13-36(5)14-16-37/h9-12,19,23,26-28,30,38,40-42H,6-8,13-18H2,1-5H3,(H,33,39)(H,34,35)/t23-,26-,27+,28-,30+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50426895
(CHEMBL2323683)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)N2CCNCC2)cc1 |r| Show InChI InChI=1S/C31H47N5O8/c1-18(2)24-21(28(35-34-24)44-29-27(41)26(40)25(39)22(17-37)43-29)16-20-10-8-19(9-11-20)6-5-7-23(38)33-31(3,4)30(42)36-14-12-32-13-15-36/h8-11,18,22,25-27,29,32,37,39-41H,5-7,12-17H2,1-4H3,(H,33,38)(H,34,35)/t22-,25-,26+,27-,29+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Rattus norvegicus) | BDBM50426887
(CHEMBL2323695)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)N2CCNCC2)cc1C |r| Show InChI InChI=1S/C32H49N5O8/c1-18(2)25-22(29(36-35-25)45-30-28(42)27(41)26(40)23(17-38)44-30)16-21-10-9-20(15-19(21)3)7-6-8-24(39)34-32(4,5)31(43)37-13-11-33-12-14-37/h9-10,15,18,23,26-28,30,33,38,40-42H,6-8,11-14,16-17H2,1-5H3,(H,34,39)(H,35,36)/t23-,26-,27+,28-,30+/m1/s1 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of rat SGLT1 |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426889
(CHEMBL2323409)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)NCCN(C)C)cc1 |r| Show InChI InChI=1S/C31H49N5O8/c1-18(2)24-21(28(35-34-24)44-29-27(41)26(40)25(39)22(17-37)43-29)16-20-12-10-19(11-13-20)8-7-9-23(38)33-31(3,4)30(42)32-14-15-36(5)6/h10-13,18,22,25-27,29,37,39-41H,7-9,14-17H2,1-6H3,(H,32,42)(H,33,38)(H,34,35)/t22-,25-,26+,27-,29+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426893
(CHEMBL2323405)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)N2CCCCC2)cc1 |r| Show InChI InChI=1S/C32H48N4O8/c1-19(2)25-22(29(35-34-25)44-30-28(41)27(40)26(39)23(18-37)43-30)17-21-13-11-20(12-14-21)9-8-10-24(38)33-32(3,4)31(42)36-15-6-5-7-16-36/h11-14,19,23,26-28,30,37,39-41H,5-10,15-18H2,1-4H3,(H,33,38)(H,34,35)/t23-,26-,27+,28-,30+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50426893
(CHEMBL2323405)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)N2CCCCC2)cc1 |r| Show InChI InChI=1S/C32H48N4O8/c1-19(2)25-22(29(35-34-25)44-30-28(41)27(40)26(39)23(18-37)43-30)17-21-13-11-20(12-14-21)9-8-10-24(38)33-32(3,4)31(42)36-15-6-5-7-16-36/h11-14,19,23,26-28,30,37,39-41H,5-10,15-18H2,1-4H3,(H,33,38)(H,34,35)/t23-,26-,27+,28-,30+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 42 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426905
(CHEMBL2323693)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(N)=O)cc1 |r| Show InChI InChI=1S/C27H40N4O8/c1-14(2)20-17(24(31-30-20)39-25-23(36)22(35)21(34)18(13-32)38-25)12-16-10-8-15(9-11-16)6-5-7-19(33)29-27(3,4)26(28)37/h8-11,14,18,21-23,25,32,34-36H,5-7,12-13H2,1-4H3,(H2,28,37)(H,29,33)(H,30,31)/t18-,21-,22+,23-,25+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 45 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50426889
(CHEMBL2323409)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)NCCN(C)C)cc1 |r| Show InChI InChI=1S/C31H49N5O8/c1-18(2)24-21(28(35-34-24)44-29-27(41)26(40)25(39)22(17-37)43-29)16-20-12-10-19(11-13-20)8-7-9-23(38)33-31(3,4)30(42)32-14-15-36(5)6/h10-13,18,22,25-27,29,37,39-41H,7-9,14-17H2,1-6H3,(H,32,42)(H,33,38)(H,34,35)/t22-,25-,26+,27-,29+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 46 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426888
(CHEMBL2323694)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)N2CCNCC2)cc1 |r| Show InChI InChI=1S/C31H47N5O8/c1-18(2)24-21(28(35-34-24)44-29-27(41)26(40)25(39)22(17-37)43-29)16-20-10-8-19(9-11-20)6-5-7-23(38)33-31(3,4)30(42)36-14-12-32-13-15-36/h8-11,18,22,25-27,29,32,37,39-41H,5-7,12-17H2,1-4H3,(H,33,38)(H,34,35)/t22-,25+,26+,27-,29+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426891
(CHEMBL2323407)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)NCCO)cc1 |r| Show InChI InChI=1S/C29H44N4O9/c1-16(2)22-19(26(33-32-22)42-27-25(39)24(38)23(37)20(15-35)41-27)14-18-10-8-17(9-11-18)6-5-7-21(36)31-29(3,4)28(40)30-12-13-34/h8-11,16,20,23-25,27,34-35,37-39H,5-7,12-15H2,1-4H3,(H,30,40)(H,31,36)(H,32,33)/t20-,23-,24+,25-,27+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50426905
(CHEMBL2323693)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(N)=O)cc1 |r| Show InChI InChI=1S/C27H40N4O8/c1-14(2)20-17(24(31-30-20)39-25-23(36)22(35)21(34)18(13-32)38-25)12-16-10-8-15(9-11-16)6-5-7-19(33)29-27(3,4)26(28)37/h8-11,14,18,21-23,25,32,34-36H,5-7,12-13H2,1-4H3,(H2,28,37)(H,29,33)(H,30,31)/t18-,21-,22+,23-,25+/m1/s1 | PDB
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| n/a | n/a | 80 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50426892
(CHEMBL2323406)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)N2CCOCC2)cc1 |r| Show InChI InChI=1S/C31H46N4O9/c1-18(2)24-21(28(34-33-24)44-29-27(40)26(39)25(38)22(17-36)43-29)16-20-10-8-19(9-11-20)6-5-7-23(37)32-31(3,4)30(41)35-12-14-42-15-13-35/h8-11,18,22,25-27,29,36,38-40H,5-7,12-17H2,1-4H3,(H,32,37)(H,33,34)/t22-,25-,26+,27-,29+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
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| n/a | n/a | 98 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426890
(CHEMBL2323408)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)NCC(N)=O)cc1 |r| Show InChI InChI=1S/C29H43N5O9/c1-15(2)22-18(26(34-33-22)43-27-25(40)24(39)23(38)19(14-35)42-27)12-17-10-8-16(9-11-17)6-5-7-21(37)32-29(3,4)28(41)31-13-20(30)36/h8-11,15,19,23-25,27,35,38-40H,5-7,12-14H2,1-4H3,(H2,30,36)(H,31,41)(H,32,37)(H,33,34)/t19-,23-,24+,25-,27+/m1/s1 | PDB
UniProtKB/SwissProt
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| n/a | n/a | 103 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Rattus norvegicus) | BDBM50426888
(CHEMBL2323694)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)N2CCNCC2)cc1 |r| Show InChI InChI=1S/C31H47N5O8/c1-18(2)24-21(28(35-34-24)44-29-27(41)26(40)25(39)22(17-37)43-29)16-20-10-8-19(9-11-20)6-5-7-23(38)33-31(3,4)30(42)36-14-12-32-13-15-36/h8-11,18,22,25-27,29,32,37,39-41H,5-7,12-17H2,1-4H3,(H,33,38)(H,34,35)/t22-,25+,26+,27-,29+/m1/s1 | PDB
Reactome pathway
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PubMed
| n/a | n/a | 104 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of rat SGLT1 |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426892
(CHEMBL2323406)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)N2CCOCC2)cc1 |r| Show InChI InChI=1S/C31H46N4O9/c1-18(2)24-21(28(34-33-24)44-29-27(40)26(39)25(38)22(17-36)43-29)16-20-10-8-19(9-11-20)6-5-7-23(37)32-31(3,4)30(41)35-12-14-42-15-13-35/h8-11,18,22,25-27,29,36,38-40H,5-7,12-17H2,1-4H3,(H,32,37)(H,33,34)/t22-,25-,26+,27-,29+/m1/s1 | PDB
UniProtKB/SwissProt
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| n/a | n/a | 124 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50426891
(CHEMBL2323407)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)NCCO)cc1 |r| Show InChI InChI=1S/C29H44N4O9/c1-16(2)22-19(26(33-32-22)42-27-25(39)24(38)23(37)20(15-35)41-27)14-18-10-8-17(9-11-18)6-5-7-21(36)31-29(3,4)28(40)30-12-13-34/h8-11,16,20,23-25,27,34-35,37-39H,5-7,12-15H2,1-4H3,(H,30,40)(H,31,36)(H,32,33)/t20-,23-,24+,25-,27+/m1/s1 | PDB
UniProtKB/SwissProt
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PubMed
| n/a | n/a | 151 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426897
(CHEMBL2323417)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NCCCO)cc1 |r| Show InChI InChI=1S/C26H39N3O8/c1-15(2)21-18(25(29-28-21)37-26-24(35)23(34)22(33)19(14-31)36-26)13-17-9-7-16(8-10-17)5-3-6-20(32)27-11-4-12-30/h7-10,15,19,22-24,26,30-31,33-35H,3-6,11-14H2,1-2H3,(H,27,32)(H,28,29)/t19-,22-,23+,24-,26+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
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| CHEMBL
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| Article
PubMed
| n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Rattus norvegicus) | BDBM50394533
(CHEMBL2159101)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(O)cc1C |r| Show InChI InChI=1S/C20H28N2O7/c1-9(2)15-13(7-11-4-5-12(24)6-10(11)3)19(22-21-15)29-20-18(27)17(26)16(25)14(8-23)28-20/h4-6,9,14,16-18,20,23-27H,7-8H2,1-3H3,(H,21,22)/t14-,16-,17+,18-,20+/m1/s1 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
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| CHEMBL
KEGG
PC cid
PC sid
UniChem
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| Article
PubMed
| n/a | n/a | 183 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of rat SGLT1 |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50394538
(CHEMBL2159106)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(O)cc1 |r| Show InChI InChI=1S/C19H26N2O7/c1-9(2)14-12(7-10-3-5-11(23)6-4-10)18(21-20-14)28-19-17(26)16(25)15(24)13(8-22)27-19/h3-6,9,13,15-17,19,22-26H,7-8H2,1-2H3,(H,20,21)/t13-,15-,16+,17-,19+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
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PubMed
| n/a | n/a | 207 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50426890
(CHEMBL2323408)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)NCC(N)=O)cc1 |r| Show InChI InChI=1S/C29H43N5O9/c1-15(2)22-18(26(34-33-22)43-27-25(40)24(39)23(38)19(14-35)42-27)12-17-10-8-16(9-11-17)6-5-7-21(37)32-29(3,4)28(41)31-13-20(30)36/h8-11,15,19,23-25,27,35,38-40H,5-7,12-14H2,1-4H3,(H2,30,36)(H,31,41)(H,32,37)(H,33,34)/t19-,23-,24+,25-,27+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
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PubMed
| n/a | n/a | 209 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426899
(CHEMBL2323415)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NCCO)cc1 |r| Show InChI InChI=1S/C25H37N3O8/c1-14(2)20-17(12-16-8-6-15(7-9-16)4-3-5-19(31)26-10-11-29)24(28-27-20)36-25-23(34)22(33)21(32)18(13-30)35-25/h6-9,14,18,21-23,25,29-30,32-34H,3-5,10-13H2,1-2H3,(H,26,31)(H,27,28)/t18-,21-,22+,23-,25+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
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| CHEMBL
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PC sid
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| Article
PubMed
| n/a | n/a | 217 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50394538
(CHEMBL2159106)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(O)cc1 |r| Show InChI InChI=1S/C19H26N2O7/c1-9(2)14-12(7-10-3-5-11(23)6-4-10)18(21-20-14)28-19-17(26)16(25)15(24)13(8-22)27-19/h3-6,9,13,15-17,19,22-26H,7-8H2,1-2H3,(H,20,21)/t13-,15-,16+,17-,19+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
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| Article
PubMed
| n/a | n/a | 285 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50426897
(CHEMBL2323417)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NCCCO)cc1 |r| Show InChI InChI=1S/C26H39N3O8/c1-15(2)21-18(25(29-28-21)37-26-24(35)23(34)22(33)19(14-31)36-26)13-17-9-7-16(8-10-17)5-3-6-20(32)27-11-4-12-30/h7-10,15,19,22-24,26,30-31,33-35H,3-6,11-14H2,1-2H3,(H,27,32)(H,28,29)/t19-,22-,23+,24-,26+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
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| CHEMBL
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PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 319 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426901
(CHEMBL2323413)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(N)=O)cc1 |r| Show InChI InChI=1S/C23H33N3O7/c1-12(2)18-15(10-14-8-6-13(7-9-14)4-3-5-17(24)28)22(26-25-18)33-23-21(31)20(30)19(29)16(11-27)32-23/h6-9,12,16,19-21,23,27,29-31H,3-5,10-11H2,1-2H3,(H2,24,28)(H,25,26)/t16-,19-,20+,21-,23+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
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PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 351 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50426898
(CHEMBL2323416)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)N(C)CCO)cc1 |r| Show InChI InChI=1S/C26H39N3O8/c1-15(2)21-18(25(28-27-21)37-26-24(35)23(34)22(33)19(14-31)36-26)13-17-9-7-16(8-10-17)5-4-6-20(32)29(3)11-12-30/h7-10,15,19,22-24,26,30-31,33-35H,4-6,11-14H2,1-3H3,(H,27,28)/t19-,22-,23+,24-,26+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
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| CHEMBL
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PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 358 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50426887
(CHEMBL2323695)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)N2CCNCC2)cc1C |r| Show InChI InChI=1S/C32H49N5O8/c1-18(2)25-22(29(36-35-25)45-30-28(42)27(41)26(40)23(17-38)44-30)16-21-10-9-20(15-19(21)3)7-6-8-24(39)34-32(4,5)31(43)37-13-11-33-12-14-37/h9-10,15,18,23,26-28,30,33,38,40-42H,6-8,11-14,16-17H2,1-5H3,(H,34,39)(H,35,36)/t23-,26-,27+,28-,30+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
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PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 371 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426912
(CHEMBL2323686)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(NC(C)=O)cc1 |r| Show InChI InChI=1S/C21H29N3O7/c1-10(2)16-14(8-12-4-6-13(7-5-12)22-11(3)26)20(24-23-16)31-21-19(29)18(28)17(27)15(9-25)30-21/h4-7,10,15,17-19,21,25,27-29H,8-9H2,1-3H3,(H,22,26)(H,23,24)/t15-,17-,18+,19-,21+/m1/s1 | PDB
UniProtKB/SwissProt
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| n/a | n/a | 392 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426913
(CHEMBL2323685)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(N)cc1 |r| Show InChI InChI=1S/C19H27N3O6/c1-9(2)14-12(7-10-3-5-11(20)6-4-10)18(22-21-14)28-19-17(26)16(25)15(24)13(8-23)27-19/h3-6,9,13,15-17,19,23-26H,7-8,20H2,1-2H3,(H,21,22)/t13-,15-,16+,17-,19+/m1/s1 | PDB
UniProtKB/SwissProt
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| n/a | n/a | 422 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426907
(CHEMBL2323691)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(NC(=O)CCN)cc1 |r| Show InChI InChI=1S/C22H32N4O7/c1-11(2)17-14(9-12-3-5-13(6-4-12)24-16(28)7-8-23)21(26-25-17)33-22-20(31)19(30)18(29)15(10-27)32-22/h3-6,11,15,18-20,22,27,29-31H,7-10,23H2,1-2H3,(H,24,28)(H,25,26)/t15-,18-,19+,20-,22+/m1/s1 | PDB
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| n/a | n/a | 446 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50426900
(CHEMBL2323414)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCCC(N)=O)cc1 |r| Show InChI InChI=1S/C24H35N3O7/c1-13(2)19-16(11-15-9-7-14(8-10-15)5-3-4-6-18(25)29)23(27-26-19)34-24-22(32)21(31)20(30)17(12-28)33-24/h7-10,13,17,20-22,24,28,30-32H,3-6,11-12H2,1-2H3,(H2,25,29)(H,26,27)/t17-,20-,21+,22-,24+/m1/s1 | PDB
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| n/a | n/a | 457 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426898
(CHEMBL2323416)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)N(C)CCO)cc1 |r| Show InChI InChI=1S/C26H39N3O8/c1-15(2)21-18(25(28-27-21)37-26-24(35)23(34)22(33)19(14-31)36-26)13-17-9-7-16(8-10-17)5-4-6-20(32)29(3)11-12-30/h7-10,15,19,22-24,26,30-31,33-35H,4-6,11-14H2,1-3H3,(H,27,28)/t19-,22-,23+,24-,26+/m1/s1 | PDB
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| n/a | n/a | 517 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50426899
(CHEMBL2323415)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NCCO)cc1 |r| Show InChI InChI=1S/C25H37N3O8/c1-14(2)20-17(12-16-8-6-15(7-9-16)4-3-5-19(31)26-10-11-29)24(28-27-20)36-25-23(34)22(33)21(32)18(13-30)35-25/h6-9,14,18,21-23,25,29-30,32-34H,3-5,10-13H2,1-2H3,(H,26,31)(H,27,28)/t18-,21-,22+,23-,25+/m1/s1 | PDB
UniProtKB/SwissProt
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| n/a | n/a | 608 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426911
(CHEMBL2323687)Show SMILES CCC(=O)Nc1ccc(Cc2c(O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)[nH]nc2C(C)C)cc1 |r| Show InChI InChI=1S/C22H31N3O7/c1-4-16(27)23-13-7-5-12(6-8-13)9-14-17(11(2)3)24-25-21(14)32-22-20(30)19(29)18(28)15(10-26)31-22/h5-8,11,15,18-20,22,26,28-30H,4,9-10H2,1-3H3,(H,23,27)(H,24,25)/t15-,18-,19+,20-,22+/m1/s1 | PDB
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PubMed
| n/a | n/a | 724 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50394550
(CHEMBL2160193)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccccc1 |r| Show InChI InChI=1S/C19H26N2O6/c1-10(2)14-12(8-11-6-4-3-5-7-11)18(21-20-14)27-19-17(25)16(24)15(23)13(9-22)26-19/h3-7,10,13,15-17,19,22-25H,8-9H2,1-2H3,(H,20,21)/t13-,15-,16+,17-,19+/m1/s1 | PDB
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| n/a | n/a | 738 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426896
(CHEMBL2323418)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NCC(N)=O)cc1 |r| Show InChI InChI=1S/C25H36N4O8/c1-13(2)20-16(24(29-28-20)37-25-23(35)22(34)21(33)17(12-30)36-25)10-15-8-6-14(7-9-15)4-3-5-19(32)27-11-18(26)31/h6-9,13,17,21-23,25,30,33-35H,3-5,10-12H2,1-2H3,(H2,26,31)(H,27,32)(H,28,29)/t17-,21-,22+,23-,25+/m1/s1 | PDB
UniProtKB/SwissProt
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PubMed
| n/a | n/a | 772 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426908
(CHEMBL2323690)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(NC(=O)CN)cc1 |r| Show InChI InChI=1S/C21H30N4O7/c1-10(2)16-13(7-11-3-5-12(6-4-11)23-15(27)8-22)20(25-24-16)32-21-19(30)18(29)17(28)14(9-26)31-21/h3-6,10,14,17-19,21,26,28-30H,7-9,22H2,1-2H3,(H,23,27)(H,24,25)/t14-,17-,18+,19-,21+/m1/s1 | PDB
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PubMed
| n/a | n/a | 831 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426909
(CHEMBL2323689)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(NS(C)(=O)=O)cc1 |r| Show InChI InChI=1S/C20H29N3O8S/c1-10(2)15-13(8-11-4-6-12(7-5-11)23-32(3,28)29)19(22-21-15)31-20-18(27)17(26)16(25)14(9-24)30-20/h4-7,10,14,16-18,20,23-27H,8-9H2,1-3H3,(H,21,22)/t14-,16-,17+,18-,20+/m1/s1 | PDB
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| Article
PubMed
| n/a | n/a | 931 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50426909
(CHEMBL2323689)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(NS(C)(=O)=O)cc1 |r| Show InChI InChI=1S/C20H29N3O8S/c1-10(2)15-13(8-11-4-6-12(7-5-11)23-32(3,28)29)19(22-21-15)31-20-18(27)17(26)16(25)14(9-24)30-20/h4-7,10,14,16-18,20,23-27H,8-9H2,1-3H3,(H,21,22)/t14-,16-,17+,18-,20+/m1/s1 | PDB
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| Article
PubMed
| n/a | n/a | 936 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426900
(CHEMBL2323414)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCCC(N)=O)cc1 |r| Show InChI InChI=1S/C24H35N3O7/c1-13(2)19-16(11-15-9-7-14(8-10-15)5-3-4-6-18(25)29)23(27-26-19)34-24-22(32)21(31)20(30)17(12-28)33-24/h7-10,13,17,20-22,24,28,30-32H,3-6,11-12H2,1-2H3,(H2,25,29)(H,26,27)/t17-,20-,21+,22-,24+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
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| CHEMBL
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PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 1.03E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50426896
(CHEMBL2323418)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NCC(N)=O)cc1 |r| Show InChI InChI=1S/C25H36N4O8/c1-13(2)20-16(24(29-28-20)37-25-23(35)22(34)21(33)17(12-30)36-25)10-15-8-6-14(7-9-15)4-3-5-19(32)27-11-18(26)31/h6-9,13,17,21-23,25,30,33-35H,3-5,10-12H2,1-2H3,(H2,26,31)(H,27,32)(H,28,29)/t17-,21-,22+,23-,25+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
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PC cid
PC sid
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Similars
| Article
PubMed
| n/a | n/a | 1.05E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50426901
(CHEMBL2323413)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(N)=O)cc1 |r| Show InChI InChI=1S/C23H33N3O7/c1-12(2)18-15(10-14-8-6-13(7-9-14)4-3-5-17(24)28)22(26-25-18)33-23-21(31)20(30)19(29)16(11-27)32-23/h6-9,12,16,19-21,23,27,29-31H,3-5,10-11H2,1-2H3,(H2,24,28)(H,25,26)/t16-,19-,20+,21-,23+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
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| CHEMBL
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PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 1.07E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Rattus norvegicus) | BDBM50426887
(CHEMBL2323695)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(CCCC(=O)NC(C)(C)C(=O)N2CCNCC2)cc1C |r| Show InChI InChI=1S/C32H49N5O8/c1-18(2)25-22(29(36-35-25)45-30-28(42)27(41)26(40)23(17-38)44-30)16-21-10-9-20(15-19(21)3)7-6-8-24(39)34-32(4,5)31(43)37-13-11-33-12-14-37/h9-10,15,18,23,26-28,30,33,38,40-42H,6-8,11-14,16-17H2,1-5H3,(H,34,39)(H,35,36)/t23-,26-,27+,28-,30+/m1/s1 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 1.16E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of rat SGLT2 |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426904
(CHEMBL2323410)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(cc1)C(N)=O |r| Show InChI InChI=1S/C20H27N3O7/c1-9(2)14-12(7-10-3-5-11(6-4-10)18(21)28)19(23-22-14)30-20-17(27)16(26)15(25)13(8-24)29-20/h3-6,9,13,15-17,20,24-27H,7-8H2,1-2H3,(H2,21,28)(H,22,23)/t13-,15-,16+,17-,20+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
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PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 1.47E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 1
(Homo sapiens (Human)) | BDBM50426910
(CHEMBL2323688)Show SMILES CCCC(=O)Nc1ccc(Cc2c(O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)[nH]nc2C(C)C)cc1 |r| Show InChI InChI=1S/C23H33N3O7/c1-4-5-17(28)24-14-8-6-13(7-9-14)10-15-18(12(2)3)25-26-22(15)33-23-21(31)20(30)19(29)16(11-27)32-23/h6-9,12,16,19-21,23,27,29-31H,4-5,10-11H2,1-3H3,(H,24,28)(H,25,26)/t16-,19-,20+,21-,23+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT1 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
Sodium/glucose cotransporter 2
(Homo sapiens (Human)) | BDBM50426913
(CHEMBL2323685)Show SMILES CC(C)c1n[nH]c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(N)cc1 |r| Show InChI InChI=1S/C19H27N3O6/c1-9(2)14-12(7-10-3-5-11(20)6-4-10)18(22-21-14)28-19-17(26)16(25)15(24)13(8-23)27-19/h3-6,9,13,15-17,19,23-26H,7-8,20H2,1-2H3,(H,21,22)/t13-,15-,16+,17-,19+/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 1.59E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kissei Pharmaceutical Company
Curated by ChEMBL
| Assay Description
Inhibition of human SGLT2 expressed in COS7 cells assessed as inhibition [14C]-AMG cellular uptake |
Bioorg Med Chem 21: 748-65 (2013)
Article DOI: 10.1016/j.bmc.2012.11.041
BindingDB Entry DOI: 10.7270/Q2445NS9 |
More data for this
Ligand-Target Pair | |
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