Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Tumor necrosis factor (Homo sapiens (Human)) | BDBM50373071![]() (CHEMBL255489) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 1.18E+4 | n/a | n/a | n/a | n/a | n/a |
The Centre for Research and Technology of Thessaly (CE.RE.TE.TH.) , 3rd km Karditsa-Mitropolis, Karditsa 43100, Greece. Curated by ChEMBL | Assay Description Binding affinity to GST-tagged human TNF-alpha by fluorescence assay in presence of 10 % MeOH as solvent | ACS Med Chem Lett 4: 137-41 (2013) Article DOI: 10.1021/ml300380h BindingDB Entry DOI: 10.7270/Q2W66N4P | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Tumor necrosis factor (Homo sapiens (Human)) | BDBM50373071![]() (CHEMBL255489) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 9.77E+3 | n/a | n/a | n/a | n/a | n/a |
The Centre for Research and Technology of Thessaly (CE.RE.TE.TH.) , 3rd km Karditsa-Mitropolis, Karditsa 43100, Greece. Curated by ChEMBL | Assay Description Binding affinity to GST-tagged human TNF-alpha by fluorescence assay in presence of 5 % MeOH as solvent | ACS Med Chem Lett 4: 137-41 (2013) Article DOI: 10.1021/ml300380h BindingDB Entry DOI: 10.7270/Q2W66N4P | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Tumor necrosis factor (Homo sapiens (Human)) | BDBM50373071![]() (CHEMBL255489) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 8.30E+3 | n/a | n/a | n/a | n/a | n/a |
The Centre for Research and Technology of Thessaly (CE.RE.TE.TH.) , 3rd km Karditsa-Mitropolis, Karditsa 43100, Greece. Curated by ChEMBL | Assay Description Binding affinity to GST-tagged human TNF-alpha by fluorescence assay in presence of 2.5 % MeOH as solvent | ACS Med Chem Lett 4: 137-41 (2013) Article DOI: 10.1021/ml300380h BindingDB Entry DOI: 10.7270/Q2W66N4P | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Tumor necrosis factor (Homo sapiens (Human)) | BDBM50373071![]() (CHEMBL255489) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 6.18E+3 | n/a | n/a | n/a | n/a | n/a |
The Centre for Research and Technology of Thessaly (CE.RE.TE.TH.) , 3rd km Karditsa-Mitropolis, Karditsa 43100, Greece. Curated by ChEMBL | Assay Description Binding affinity to GST-tagged human TNF-alpha by fluorescence assay in presence of 5 % PEG3350 as solvent | ACS Med Chem Lett 4: 137-41 (2013) Article DOI: 10.1021/ml300380h BindingDB Entry DOI: 10.7270/Q2W66N4P | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Tumor necrosis factor (Homo sapiens (Human)) | BDBM50373071![]() (CHEMBL255489) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 5.36E+3 | n/a | n/a | n/a | n/a | n/a |
The Centre for Research and Technology of Thessaly (CE.RE.TE.TH.) , 3rd km Karditsa-Mitropolis, Karditsa 43100, Greece. Curated by ChEMBL | Assay Description Binding affinity to GST-tagged human TNF-alpha by fluorescence assay in presence of 5 % DMSO as solvent | ACS Med Chem Lett 4: 137-41 (2013) Article DOI: 10.1021/ml300380h BindingDB Entry DOI: 10.7270/Q2W66N4P | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Tumor necrosis factor (Homo sapiens (Human)) | BDBM50373071![]() (CHEMBL255489) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 5.36E+3 | n/a | n/a | n/a | 6.5 | n/a |
The Centre for Research and Technology of Thessaly (CE.RE.TE.TH.) , 3rd km Karditsa-Mitropolis, Karditsa 43100, Greece. Curated by ChEMBL | Assay Description Binding affinity to GST-tagged human TNF-alpha in 10 mM citrate-phosphate at pH 6.5 by fluorescence assay | ACS Med Chem Lett 4: 137-41 (2013) Article DOI: 10.1021/ml300380h BindingDB Entry DOI: 10.7270/Q2W66N4P | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Tumor necrosis factor (Homo sapiens (Human)) | BDBM50373071![]() (CHEMBL255489) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 5.75E+3 | n/a | n/a | n/a | n/a | n/a |
The Centre for Research and Technology of Thessaly (CE.RE.TE.TH.) , 3rd km Karditsa-Mitropolis, Karditsa 43100, Greece. Curated by ChEMBL | Assay Description Binding affinity to GST-tagged human TNF-alpha by fluorescence assay in presence of 2.5 % PEG3350 as solvent | ACS Med Chem Lett 4: 137-41 (2013) Article DOI: 10.1021/ml300380h BindingDB Entry DOI: 10.7270/Q2W66N4P | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Tumor necrosis factor (Homo sapiens (Human)) | BDBM50373071![]() (CHEMBL255489) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 7.51E+3 | n/a | n/a | n/a | n/a | n/a |
The Centre for Research and Technology of Thessaly (CE.RE.TE.TH.) , 3rd km Karditsa-Mitropolis, Karditsa 43100, Greece. Curated by ChEMBL | Assay Description Binding affinity to GST-tagged human TNF-alpha by fluorescence assay in presence of 2.5 % DMF as solvent | ACS Med Chem Lett 4: 137-41 (2013) Article DOI: 10.1021/ml300380h BindingDB Entry DOI: 10.7270/Q2W66N4P | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Tumor necrosis factor (Homo sapiens (Human)) | BDBM50373071![]() (CHEMBL255489) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 7.34E+3 | n/a | n/a | n/a | n/a | n/a |
The Centre for Research and Technology of Thessaly (CE.RE.TE.TH.) , 3rd km Karditsa-Mitropolis, Karditsa 43100, Greece. Curated by ChEMBL | Assay Description Binding affinity to GST-tagged human TNF-alpha by fluorescence assay in presence of 10 % DMSO as solvent | ACS Med Chem Lett 4: 137-41 (2013) Article DOI: 10.1021/ml300380h BindingDB Entry DOI: 10.7270/Q2W66N4P | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Tumor necrosis factor (Homo sapiens (Human)) | BDBM50373071![]() (CHEMBL255489) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 5.70E+3 | n/a | n/a | n/a | n/a | n/a |
The Centre for Research and Technology of Thessaly (CE.RE.TE.TH.) , 3rd km Karditsa-Mitropolis, Karditsa 43100, Greece. Curated by ChEMBL | Assay Description Binding affinity to GST-tagged human TNF-alpha by fluorescence assay in presence of 2.5 % DMSO as solvent | ACS Med Chem Lett 4: 137-41 (2013) Article DOI: 10.1021/ml300380h BindingDB Entry DOI: 10.7270/Q2W66N4P | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Tumor necrosis factor (Homo sapiens (Human)) | BDBM50373071![]() (CHEMBL255489) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 8.44E+3 | n/a | n/a | n/a | n/a | n/a |
The Centre for Research and Technology of Thessaly (CE.RE.TE.TH.) , 3rd km Karditsa-Mitropolis, Karditsa 43100, Greece. Curated by ChEMBL | Assay Description Binding affinity to GST-tagged human TNF-alpha by fluorescence assay in presence of 10 % PEG3350 as solvent | ACS Med Chem Lett 4: 137-41 (2013) Article DOI: 10.1021/ml300380h BindingDB Entry DOI: 10.7270/Q2W66N4P | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) |