Found 35 hits Enz. Inhib. hit(s) with all data for entry = 50043452 Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Glucagon receptor
(Homo sapiens (Human)) | BDBM50071873
(4-[2-(4-Fluoro-phenyl)-5-(4-methanesulfinyl-phenyl...)Show SMILES CS(=O)c1ccc(cc1)-c1cc(c([nH]1)-c1ccc(F)cc1)-c1ccncc1 Show InChI InChI=1S/C22H17FN2OS/c1-27(26)19-8-4-16(5-9-19)21-14-20(15-10-12-24-13-11-15)22(25-21)17-2-6-18(23)7-3-17/h2-14,25H,1H3 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet 
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| Article
| n/a | n/a | 5.30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM13336
(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)Show SMILES CS(=O)c1ccc(cc1)-c1nc(c([nH]1)-c1ccc(F)cc1)-c1ccncc1 Show InChI InChI=1S/C21H16FN3OS/c1-27(26)18-8-4-16(5-9-18)21-24-19(14-2-6-17(22)7-3-14)20(25-21)15-10-12-23-13-11-15/h2-13H,1H3,(H,24,25) | PDB
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UniProtKB/SwissProt
B.MOAD
antibodypedia
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| Purchase
CHEMBL
MMDB
PC cid
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PDB
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| Article
| n/a | n/a | 37 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50071894
(4-[2-(4-Fluoro-phenyl)-5-(4-methylsulfanyl-phenyl)...)Show SMILES CSc1ccc(cc1)-c1cc(c([nH]1)-c1ccc(F)cc1)-c1ccncc1 Show InChI InChI=1S/C22H17FN2S/c1-26-19-8-4-16(5-9-19)21-14-20(15-10-12-24-13-11-15)22(25-21)17-2-6-18(23)7-3-17/h2-14,25H,1H3 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
| n/a | n/a | 44 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075751
(4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-1H-pyrrol-2-...)Show SMILES Fc1ccc(cc1)-c1cc([nH]c1-c1ccncc1)-c1ccc(cc1)C#N Show InChI InChI=1S/C22H14FN3/c23-19-7-5-16(6-8-19)20-13-21(17-3-1-15(14-24)2-4-17)26-22(20)18-9-11-25-12-10-18/h1-13,26H | PDB
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UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
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| Article
| n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075794
(4-[3-(4-Fluoro-phenyl)-5-(4-nitro-phenyl)-1H-pyrro...)Show SMILES [O-][N+](=O)c1ccc(cc1)-c1cc(c([nH]1)-c1ccncc1)-c1ccc(F)cc1 Show InChI InChI=1S/C21H14FN3O2/c22-17-5-1-14(2-6-17)19-13-20(15-3-7-18(8-4-15)25(26)27)24-21(19)16-9-11-23-12-10-16/h1-13,24H | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
| n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075767
(4-[3-(3-Bromo-phenyl)-5-(4-chloro-phenyl)-1H-pyrro...)Show SMILES Clc1ccc(cc1)-c1cc(c([nH]1)-c1ccncc1)-c1cccc(Br)c1 Show InChI InChI=1S/C21H14BrClN2/c22-17-3-1-2-16(12-17)19-13-20(14-4-6-18(23)7-5-14)25-21(19)15-8-10-24-11-9-15/h1-13,25H | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
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| Article
| n/a | n/a | 80 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075782
(4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-1H-pyrrol-2-...)Show SMILES OC(=O)c1ccc(cc1)-c1cc(c([nH]1)-c1ccncc1)-c1ccc(F)cc1 Show InChI InChI=1S/C22H15FN2O2/c23-18-7-5-14(6-8-18)19-13-20(15-1-3-17(4-2-15)22(26)27)25-21(19)16-9-11-24-12-10-16/h1-13,25H,(H,26,27) | PDB
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B.MOAD
antibodypedia
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| CHEMBL
PC cid
PC sid
UniChem
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| Article
| n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075778
(4-[5-(4-Fluoro-phenyl)-2-(4-methylsulfanyl-phenyl)...)Show SMILES CSc1ccc(cc1)-c1nc(c([nH]1)-c1ccc(F)cc1)-c1ccncc1 Show InChI InChI=1S/C21H16FN3S/c1-26-18-8-4-16(5-9-18)21-24-19(14-2-6-17(22)7-3-14)20(25-21)15-10-12-23-13-11-15/h2-13H,1H3,(H,24,25) | PDB
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antibodypedia
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| Purchase
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| Article
| n/a | n/a | 117 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075764
(4-[3,5-Bis-(4-chloro-phenyl)-1H-pyrrol-2-yl]-pyrid...)Show SMILES Clc1ccc(cc1)-c1cc(c([nH]1)-c1ccncc1)-c1ccc(Cl)cc1 Show InChI InChI=1S/C21H14Cl2N2/c22-17-5-1-14(2-6-17)19-13-20(15-3-7-18(23)8-4-15)25-21(19)16-9-11-24-12-10-16/h1-13,25H | PDB
MMDB
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B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
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| Article
| n/a | n/a | 160 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075789
(4-[3-(4-Fluoro-phenyl)-1H-pyrrol-2-yl]-pyridine | ...)Show InChI InChI=1S/C15H11FN2/c16-13-3-1-11(2-4-13)14-7-10-18-15(14)12-5-8-17-9-6-12/h1-10,18H | PDB
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B.MOAD
antibodypedia
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AffyNet
| CHEMBL
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UniChem
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| Article
| n/a | n/a | 160 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075769
(4-[5-Cyclohexyl-3-(4-fluoro-phenyl)-1H-pyrrol-2-yl...)Show InChI InChI=1S/C21H21FN2/c22-18-8-6-15(7-9-18)19-14-20(16-4-2-1-3-5-16)24-21(19)17-10-12-23-13-11-17/h6-14,16,24H,1-5H2 | PDB
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| CHEMBL
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| Article
| n/a | n/a | 180 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075776
(4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-1H-pyrrol-2-...)Show SMILES Nc1ccc(cc1)-c1cc(c([nH]1)-c1ccncc1)-c1ccc(F)cc1 Show InChI InChI=1S/C21H16FN3/c22-17-5-1-14(2-6-17)19-13-20(15-3-7-18(23)8-4-15)25-21(19)16-9-11-24-12-10-16/h1-13,25H,23H2 | PDB
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antibodypedia
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| CHEMBL
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PC sid
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| Article
| n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075774
(4-[5-(4-Chloro-phenyl)-3-phenyl-1H-pyrrol-2-yl]-py...)Show SMILES Clc1ccc(cc1)-c1cc(c([nH]1)-c1ccncc1)-c1ccccc1 Show InChI InChI=1S/C21H15ClN2/c22-18-8-6-16(7-9-18)20-14-19(15-4-2-1-3-5-15)21(24-20)17-10-12-23-13-11-17/h1-14,24H | PDB
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UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
| n/a | n/a | 210 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075785
(4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-1H-pyrrol-2-...)Show SMILES CCOC(=O)c1ccc(cc1)-c1cc(c([nH]1)-c1ccncc1)-c1ccc(F)cc1 Show InChI InChI=1S/C24H19FN2O2/c1-2-29-24(28)19-5-3-17(4-6-19)22-15-21(16-7-9-20(25)10-8-16)23(27-22)18-11-13-26-14-12-18/h3-15,27H,2H2,1H3 | PDB
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| CHEMBL
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PC sid
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| Article
| n/a | n/a | 260 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075777
(4-[3-(4-Bromo-phenyl)-5-(4-chloro-phenyl)-1H-pyrro...)Show SMILES Clc1ccc(cc1)-c1cc(c([nH]1)-c1ccncc1)-c1ccc(Br)cc1 Show InChI InChI=1S/C21H14BrClN2/c22-17-5-1-14(2-6-17)19-13-20(15-3-7-18(23)8-4-15)25-21(19)16-9-11-24-12-10-16/h1-13,25H | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
| n/a | n/a | 301 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075779
(4-[3-(4-Fluoro-phenyl)-5-methyl-1H-pyrrol-2-yl]-py...)Show InChI InChI=1S/C16H13FN2/c1-11-10-15(12-2-4-14(17)5-3-12)16(19-11)13-6-8-18-9-7-13/h2-10,19H,1H3 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
| n/a | n/a | 321 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075753
(4-[3,5-Bis-(4-fluoro-phenyl)-1H-pyrrol-2-yl]-pyrid...)Show SMILES Fc1ccc(cc1)-c1cc(c([nH]1)-c1ccncc1)-c1ccc(F)cc1 Show InChI InChI=1S/C21H14F2N2/c22-17-5-1-14(2-6-17)19-13-20(15-3-7-18(23)8-4-15)25-21(19)16-9-11-24-12-10-16/h1-13,25H | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
| n/a | n/a | 340 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075760
(4-[5-(4-Chloro-phenyl)-3-(3-methoxy-phenyl)-1H-pyr...)Show SMILES COc1cccc(c1)-c1cc([nH]c1-c1ccncc1)-c1ccc(Cl)cc1 Show InChI InChI=1S/C22H17ClN2O/c1-26-19-4-2-3-17(13-19)20-14-21(15-5-7-18(23)8-6-15)25-22(20)16-9-11-24-12-10-16/h2-14,25H,1H3 | PDB
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B.MOAD
antibodypedia
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AffyNet
| CHEMBL
PC cid
PC sid
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| Article
| n/a | n/a | 421 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075757
(4-[5-(2,4-Dichloro-phenyl)-3-(4-fluoro-phenyl)-1H-...)Show SMILES Fc1ccc(cc1)-c1cc([nH]c1-c1ccncc1)-c1ccc(Cl)cc1Cl Show InChI InChI=1S/C21H13Cl2FN2/c22-15-3-6-17(19(23)11-15)20-12-18(13-1-4-16(24)5-2-13)21(26-20)14-7-9-25-10-8-14/h1-12,26H | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
| n/a | n/a | 421 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075788
(4-[5-(3-Chloro-phenyl)-3-(4-fluoro-phenyl)-1H-pyrr...)Show SMILES Fc1ccc(cc1)-c1cc([nH]c1-c1ccncc1)-c1cccc(Cl)c1 Show InChI InChI=1S/C21H14ClFN2/c22-17-3-1-2-16(12-17)20-13-19(14-4-6-18(23)7-5-14)21(25-20)15-8-10-24-11-9-15/h1-13,25H | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
| n/a | n/a | 421 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075756
(4-(3-(4-fluorophenyl)-5-(4-(methylsulfinyl)phenyl)...)Show SMILES CS(=O)c1ccc(cc1)-c1cc(c([nH]1)-c1ccncc1)-c1ccc(F)cc1 Show InChI InChI=1S/C22H17FN2OS/c1-27(26)19-8-4-16(5-9-19)21-14-20(15-2-6-18(23)7-3-15)22(25-21)17-10-12-24-13-11-17/h2-14,25H,1H3 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| Article
| n/a | n/a | 671 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075762
(4-[3-(4-Fluoro-phenyl)-5-phenyl-1H-pyrrol-2-yl]-py...)Show InChI InChI=1S/C21H15FN2/c22-18-8-6-15(7-9-18)19-14-20(16-4-2-1-3-5-16)24-21(19)17-10-12-23-13-11-17/h1-14,24H | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
| n/a | n/a | 802 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075765
(4-[3-(2-Bromo-phenyl)-5-(4-chloro-phenyl)-1H-pyrro...)Show SMILES Clc1ccc(cc1)-c1cc(c([nH]1)-c1ccncc1)-c1ccccc1Br Show InChI InChI=1S/C21H14BrClN2/c22-19-4-2-1-3-17(19)18-13-20(14-5-7-16(23)8-6-14)25-21(18)15-9-11-24-12-10-15/h1-13,25H | PDB
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| Article
| n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075758
(4-[5-(4-Chloro-phenyl)-3-(4-methoxy-phenyl)-1H-pyr...)Show SMILES COc1ccc(cc1)-c1cc([nH]c1-c1ccncc1)-c1ccc(Cl)cc1 Show InChI InChI=1S/C22H17ClN2O/c1-26-19-8-4-15(5-9-19)20-14-21(16-2-6-18(23)7-3-16)25-22(20)17-10-12-24-13-11-17/h2-14,25H,1H3 | PDB
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| n/a | n/a | 1.15E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075792
(4-[3-(4-Fluoro-phenyl)-5-(4-methylsulfanyl-phenyl)...)Show SMILES CSc1ccc(cc1)-c1cc(c([nH]1)-c1ccncc1)-c1ccc(F)cc1 Show InChI InChI=1S/C22H17FN2S/c1-26-19-8-4-16(5-9-19)21-14-20(15-2-6-18(23)7-3-15)22(25-21)17-10-12-24-13-11-17/h2-14,25H,1H3 | PDB
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| n/a | n/a | 1.23E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075768
(4-[5-(4-Ethyl-phenyl)-3-(4-fluoro-phenyl)-1H-pyrro...)Show SMILES CCc1ccc(cc1)-c1cc(c([nH]1)-c1ccncc1)-c1ccc(F)cc1 Show InChI InChI=1S/C23H19FN2/c1-2-16-3-5-18(6-4-16)22-15-21(17-7-9-20(24)10-8-17)23(26-22)19-11-13-25-14-12-19/h3-15,26H,2H2,1H3 | PDB
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| n/a | n/a | 1.36E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50071899
(4-[5-(4-Chloro-phenyl)-3-(4-fluoro-phenyl)-1H-pyrr...)Show SMILES Fc1ccc(cc1)-c1cc([nH]c1-c1ccncc1)-c1ccc(Cl)cc1 Show InChI InChI=1S/C21H14ClFN2/c22-17-5-1-15(2-6-17)20-13-19(14-3-7-18(23)8-4-14)21(25-20)16-9-11-24-12-10-16/h1-13,25H | PDB
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| n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075775
(4-[3-(5-Bromo-2-propoxy-phenyl)-5-(4-chloro-phenyl...)Show SMILES CCCOc1ccc(Br)cc1-c1cc([nH]c1-c1ccncc1)-c1ccc(Cl)cc1 Show InChI InChI=1S/C24H20BrClN2O/c1-2-13-29-23-8-5-18(25)14-20(23)21-15-22(16-3-6-19(26)7-4-16)28-24(21)17-9-11-27-12-10-17/h3-12,14-15,28H,2,13H2,1H3 | PDB
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| Article
| n/a | n/a | 1.44E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075761
(4-[3-(4-Fluoro-phenyl)-5-p-tolyl-1H-pyrrol-2-yl]-p...)Show SMILES Cc1ccc(cc1)-c1cc(c([nH]1)-c1ccncc1)-c1ccc(F)cc1 Show InChI InChI=1S/C22H17FN2/c1-15-2-4-17(5-3-15)21-14-20(16-6-8-19(23)9-7-16)22(25-21)18-10-12-24-13-11-18/h2-14,25H,1H3 | PDB
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| n/a | n/a | 1.69E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075786
(4-[5-(4-Chloro-phenyl)-3-(2-methoxy-phenyl)-1H-pyr...)Show SMILES COc1ccccc1-c1cc([nH]c1-c1ccncc1)-c1ccc(Cl)cc1 Show InChI InChI=1S/C22H17ClN2O/c1-26-21-5-3-2-4-18(21)19-14-20(15-6-8-17(23)9-7-15)25-22(19)16-10-12-24-13-11-16/h2-14,25H,1H3 | PDB
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| n/a | n/a | 2.66E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075770
(4-[3-(4-Fluoro-phenyl)-5-(4-methoxy-phenyl)-1H-pyr...)Show SMILES COc1ccc(cc1)-c1cc(c([nH]1)-c1ccncc1)-c1ccc(F)cc1 Show InChI InChI=1S/C22H17FN2O/c1-26-19-8-4-16(5-9-19)21-14-20(15-2-6-18(23)7-3-15)22(25-21)17-10-12-24-13-11-17/h2-14,25H,1H3 | PDB
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| n/a | n/a | 2.81E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075766
(4-[5-(4-Chloro-phenyl)-3-(2-propoxy-phenyl)-1H-pyr...)Show SMILES CCCOc1ccccc1-c1cc([nH]c1-c1ccncc1)-c1ccc(Cl)cc1 Show InChI InChI=1S/C24H21ClN2O/c1-2-15-28-23-6-4-3-5-20(23)21-16-22(17-7-9-19(25)10-8-17)27-24(21)18-11-13-26-14-12-18/h3-14,16,27H,2,15H2,1H3 | PDB
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| n/a | n/a | 2.84E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075752
(4-[5-(4-Chloro-phenyl)-3-(2-isobutoxy-phenyl)-1H-p...)Show SMILES CC(C)COc1ccccc1-c1cc([nH]c1-c1ccncc1)-c1ccc(Cl)cc1 Show InChI InChI=1S/C25H23ClN2O/c1-17(2)16-29-24-6-4-3-5-21(24)22-15-23(18-7-9-20(26)10-8-18)28-25(22)19-11-13-27-14-12-19/h3-15,17,28H,16H2,1-2H3 | PDB
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| n/a | n/a | 3.77E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075749
(4-[3-(2-Allyloxy-phenyl)-5-(4-chloro-phenyl)-1H-py...)Show SMILES Clc1ccc(cc1)-c1cc(c([nH]1)-c1ccncc1)-c1ccccc1OCC=C Show InChI InChI=1S/C24H19ClN2O/c1-2-15-28-23-6-4-3-5-20(23)21-16-22(17-7-9-19(25)10-8-17)27-24(21)18-11-13-26-14-12-18/h2-14,16,27H,1,15H2 | PDB
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| n/a | n/a | 4.74E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
Glucagon receptor
(Homo sapiens (Human)) | BDBM50075754
(4-[5-(4-Chloro-phenyl)-3-(2-ethoxy-phenyl)-1H-pyrr...)Show SMILES CCOc1ccccc1-c1cc([nH]c1-c1ccncc1)-c1ccc(Cl)cc1 Show InChI InChI=1S/C23H19ClN2O/c1-2-27-22-6-4-3-5-19(22)20-15-21(16-7-9-18(24)10-8-16)26-23(20)17-11-13-25-14-12-17/h3-15,26H,2H2,1H3 | PDB
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| n/a | n/a | 1.42E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Antagonist activity at human glucagon receptor |
Citation and Details
Article DOI: 10.1007/s00044-013-0801-3
BindingDB Entry DOI: 10.7270/Q20G3MM3 |
More data for this
Ligand-Target Pair | |
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