Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105928![]() (CHEMBL3598047) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50106011![]() (CHEMBL3598077) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105992![]() (CHEMBL3598061) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105981![]() (CHEMBL3598052) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105930![]() (CHEMBL3598049) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105982![]() (CHEMBL3598053) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105988![]() (CHEMBL3598056) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105933![]() (CHEMBL3598051) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 4.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105985![]() (CHEMBL3598055) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105990![]() (CHEMBL3598057) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50106002![]() (CHEMBL3598070) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50106003![]() (CHEMBL3598071) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105995![]() (CHEMBL3598063) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50106009![]() (CHEMBL3598076) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50106007![]() (CHEMBL3598074) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50106008![]() (CHEMBL3598075) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105929![]() (CHEMBL3598048) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105984![]() (CHEMBL3598054) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 9.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105998![]() (CHEMBL3598065) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105991![]() (CHEMBL3598060) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105932![]() (CHEMBL3598050) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50106004![]() (CHEMBL3598072) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105997![]() (CHEMBL3598064) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105925![]() (CHEMBL3598044) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50106000![]() (CHEMBL3598066) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50106001![]() (CHEMBL3598068) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105924![]() (CHEMBL3598043) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 26 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105919![]() (CHEMBL3596632) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 29 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105922![]() (CHEMBL3598041) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 38 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50106005![]() (CHEMBL3598073) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105927![]() (CHEMBL3598046) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 54 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105993![]() (CHEMBL3598062) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105926![]() (CHEMBL3598045) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 76 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105920![]() (CHEMBL3598040) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105921![]() (CHEMBL3596216) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 530 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105923![]() (CHEMBL3598042) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 610 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50106013![]() (CHEMBL3598079) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50106012![]() (CHEMBL3598078) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo... | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105919![]() (CHEMBL3596632) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 98 | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assay | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105920![]() (CHEMBL3598040) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 570 | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assay | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105921![]() (CHEMBL3596216) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assay | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105922![]() (CHEMBL3598041) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 160 | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assay | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105923![]() (CHEMBL3598042) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assay | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105924![]() (CHEMBL3598043) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 160 | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assay | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105925![]() (CHEMBL3598044) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 30 | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assay | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105926![]() (CHEMBL3598045) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 180 | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assay | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105927![]() (CHEMBL3598046) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 130 | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assay | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105928![]() (CHEMBL3598047) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 8.10 | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assay | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105929![]() (CHEMBL3598048) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 18 | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assay | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nuclear receptor ROR-gamma (Homo sapiens (Human)) | BDBM50105930![]() (CHEMBL3598049) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6 | n/a | n/a | n/a | n/a |
Biogen Curated by ChEMBL | Assay Description Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assay | Bioorg Med Chem Lett 25: 2985-90 (2015) Article DOI: 10.1016/j.bmcl.2015.05.028 BindingDB Entry DOI: 10.7270/Q2X3508H | |||||||||||
More data for this Ligand-Target Pair |
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