Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Ataxin-1 (Homo sapiens (Human)) | BDBM481932 (US10913745, Example 8.09) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481920 (US10913745, Example 7.01) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481899 (US10913745, Example 1.13 | US10913745, Example 1.1...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481899 (US10913745, Example 1.13 | US10913745, Example 1.1...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM50187688 (CHEMBL3828650 | US10913745, Example 1.11) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481930 (US10913745, Example 8.07) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481931 (US10913745, Example 8.08) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481911 (US10913745, Example 1.25) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481896 (US10913745, Example 1.10) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481929 (US10913745, Example 8.06) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481921 (US10913745, Example 7.02) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481905 (US10913745, Example 1.19) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481922 (US10913745, Example 7.03) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481909 (US10913745, Example 1.23) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481891 (US10913745, Example 1.05) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481933 ((−)-trans-3,5-Dichlorobenzyl 2-(4-sulfamoylb...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481934 ((−)-trans-3,5-Dichlorobenzyl 2-(4-sulfamoylb...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481926 (US10913745, Example 8.03) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481908 (US10913745, Example 1.22) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 7 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481889 (US10913745, Example 1.03) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 7 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481924 (US10913745, Example 8.01) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 7.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481890 (US10913745, Example 1.04) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481923 (4-{(3aR,6aR)-5-[3-(4-Trifluoromethoxy-phenyl)-prop...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 8.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481912 (US10913745, Example 1.26) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481910 (US10913745, Example 1.24) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481904 (US10913745, Example 1.18) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481925 (US10913745, Example 8.02) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481919 ((3aS,6aS)-5-(4-Sulfamoyl-benzoyl)-hexahydro-pyrrol...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 14.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481906 (US10913745, Example 1.20) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481903 (US10913745, Example 1.17) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481915 ((3aR,6aS)-3,5-Dichlorobenzyl 5-(4-sulfamoylphenyls...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 31 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481901 (US10913745, Example 1.15) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 58.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481900 (US10913745, Example 1.14) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 64 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481928 (US10913745, Example 8.05) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 93 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481895 (US10913745, Example 1.09) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 118 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481907 (US10913745, Example 1.21) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 118 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481927 (US10913745, Example 8.04) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 166 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481892 (US10913745, Example 1.06) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 255 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481887 (US10913745, Example 1.01) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 293 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481913 ((3aR,6aS)-3,5-Dichlorobenzyl 5-(4-acetamidobenzoyl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 342 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481898 (US10913745, Example 1.12) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 440 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481888 (US10913745, Example 1.02) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 444 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481916 ((3aR,6aS)-3,5-Dichlorobenzyl 5-(4-(1H-tetrazol-5-y...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 573 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481918 ((3aR,6aS)-3,5-Dichlorobenzyl 5-(5-(methylsulfonami...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 622 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481886 ((3aR,6aS)-3,5-Dichlorobenzyl 5-(4-(N-methylsulfamo...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.16E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481894 (US10913745, Example 1.08) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481917 (4-((3aR,6aS)-5-((3,5-Dichlorobenzyloxy)carbonyl)oc...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.34E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481913 ((3aR,6aS)-3,5-Dichlorobenzyl 5-(4-acetamidobenzoyl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ataxin-1 (Homo sapiens (Human)) | BDBM481893 (US10913745, Example 1.07) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.11E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. US Patent | Assay Description Assay buffer (50 mM Tris-HCl, 140 mM NaCl, 5 mM KCl, 1 mM CaCl2, 1 mM MgCl2, 0.01% Triton-X-100, pH 8.0;ATX solution: ATX (human His-tagged) stock so... | US Patent US10913745 (2021) BindingDB Entry DOI: 10.7270/Q2NP27HS | |||||||||||
More data for this Ligand-Target Pair |