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Found 1 hit Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2A' and Ligand = 'BDBM50031922'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
5-hydroxytryptamine receptor 2A


(Rattus norvegicus (rat))		BDBM50031922
PNG
(6-Piperazin-1-yl-benzo[k]phenanthridine | CHEMBL61...)
Show SMILES C1CN(CCN1)c1nc2ccccc2c2c1ccc1ccccc21
Show InChI InChI=1S/C21H19N3/c1-2-6-16-15(5-1)9-10-18-20(16)17-7-3-4-8-19(17)23-21(18)24-13-11-22-12-14-24/h1-10,22H,11-14H2
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Similars
PubMed
 1.10E+3n/an/an/an/an/an/an/an/a



Universit£ di Siena

Curated by ChEMBL


Assay Description
Binding affinity to 5-hydroxytryptamine 2A receptor from rat cortex assayed using [3H]ketanserin as radioligand.

J Med Chem 38: 2692-704 (1995)


BindingDB Entry DOI: 10.7270/Q27H1K7H
More data for this
Ligand-Target Pair