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Found 1 hit Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2C' and Ligand = 'BDBM50010597'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
5-hydroxytryptamine receptor 2C


(Rattus norvegicus (Rat))		BDBM50010597
PNG
(1-(5-Isopropylidene-5H-dibenzo[a,d]cyclohepten-10-...)
Show SMILES [#6]-[#7]-1-[#6]-[#6]-[#7](-[#6]-[#6]-1)-[#6]-1=[#6]-c2ccccc2\[#6](=[#6](\[#6])-[#6])-c2ccccc-12 |t:8|
Show InChI InChI=1S/C23H26N2/c1-17(2)23-19-9-5-4-8-18(19)16-22(20-10-6-7-11-21(20)23)25-14-12-24(3)13-15-25/h4-11,16H,12-15H2,1-3H3
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PC cid
PC sid
UniChem

Similars
PubMed
 390n/an/an/an/an/an/an/an/a



Vanderbilt University

Curated by ChEMBL


Assay Description
Affinity of the compound was evaluated by inhibition of [125I]-LSD binding to NIH 3T3 cells transfected with cloned rat 5-hydroxytryptamine 2C recept...

J Med Chem 37: 2686-96 (1994)


BindingDB Entry DOI: 10.7270/Q28051NX
More data for this
Ligand-Target Pair