Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
5-hydroxytryptamine receptor 4 (GUINEA PIG) | BDBM50000483![]() ((BRL 43694)1-Methyl-1H-indazole-3-carboxylic acid ...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL DrugBank PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad de Alcal£ Curated by ChEMBL | Assay Description Binding affinity towards 5-HT3 receptor in rat was evaluated | Bioorg Med Chem Lett 12: 189-92 (2001) BindingDB Entry DOI: 10.7270/Q20R9PX0 | |||||||||||
More data for this Ligand-Target Pair |