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Found 1 hit Enz. Inhib. hit(s) with Target = 'ADP-ribosylhydrolase ARH3' and Ligand = 'BDBM370973'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
ADP-ribosylhydrolase ARH3


(Homo sapiens (Human))		BDBM370973
PNG
(US10239843, Example 80)
Show SMILES Cn1c(nc2ccc(cc2c1=O)S(=O)(=O)NC1(C)CC1)C1CC1
Show InChI InChI=1S/C16H19N3O3S/c1-16(7-8-16)18-23(21,22)11-5-6-13-12(9-11)15(20)19(2)14(17-13)10-3-4-10/h5-6,9-10,18H,3-4,7-8H2,1-2H3
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a>1.50E+5n/an/an/an/an/an/a



Istituto Superiore di Sanita



Assay Description
ARH3 In vitro selectivity assays were conducted in a total volume of 15 ul in a standard 384 well format. 5 ul of Human Full Length ARH3 (Enzo Life S...

J Med Chem 51: 1058-62 (2008)


BindingDB Entry DOI: 10.7270/Q21R6SSM
More data for this
Ligand-Target Pair