Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
ATP-binding cassette sub-family C member 8/ATP-sensitive inward rectifier potassium channel 11 (Homo sapiens (Human)) | BDBM50139709![]() (3-(2,4-Bis-trifluoromethyl-phenyl)-4-nitro-5-trifl...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | n/a | 540 | n/a | n/a | n/a | n/a |
GlaxoSmithKline Research & Development Curated by ChEMBL | Assay Description Maximum activation of human KATP (SUR1/Kir6.2) channel expressed in Xenopus oocytes | Bioorg Med Chem Lett 14: 813-6 (2004) BindingDB Entry DOI: 10.7270/Q29P312R | |||||||||||
More data for this Ligand-Target Pair |