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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Amine oxidase [flavin-containing] A' and Ligand = 'BDBM118196'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Amine oxidase [flavin-containing] A


(Homo sapiens (Human))		BDBM118196
PNG
(US8673966, N-(4-(7-((1-methyl-1H-imidazol-5-yl)eth...)
Show SMILES Cn1cncc1C#Cc1ccc2c(c1)occ(-c1ccc(CNS(=O)=O)cc1)c2=O
Show InChI InChI=1S/C22H17N3O4S/c1-25-14-23-12-18(25)8-4-15-5-9-19-21(10-15)29-13-20(22(19)26)17-6-2-16(3-7-17)11-24-30(27)28/h2-3,5-7,9-10,12-14,30H,11H2,1H3,(H,24,27,28)
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a>1.30E+5n/an/an/an/a7.5n/a



Gilead Sciences, Inc.

US Patent


Assay Description
MAO assays included luminogenic MAO substrate, reaction buffers, Luciferin Detection and the reconstitution buffer with esterase. Standard MAO reacti...

US Patent US8673966 (2014)


BindingDB Entry DOI: 10.7270/Q2QZ28MX
More data for this
Ligand-Target Pair