Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50276157 (Alternariol 5-O-Methyl Ether | CHEMBL483526) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | 340 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50276157 (Alternariol 5-O-Methyl Ether | CHEMBL483526) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | n/a | n/a | 1.71E+3 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50276157 (Alternariol 5-O-Methyl Ether | CHEMBL483526) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.71E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sunchon National University Curated by ChEMBL | Assay Description Inhibition of recombinant human MAO-A using kynuramine as substrate incubated for 10 mins by spectrophotometric method | Bioorg Med Chem Lett 28: 2403-2407 (2018) Article DOI: 10.1016/j.bmcl.2018.06.023 BindingDB Entry DOI: 10.7270/Q23R0WCT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50276157 (Alternariol 5-O-Methyl Ether | CHEMBL483526) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.71E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sunchon National University Curated by ChEMBL | Assay Description Inhibition of human recombinant MAOA using kynuramine as substrate preincubated for 30 mins followed by substrate addition | Bioorg Med Chem Lett 28: 584-588 (2018) Article DOI: 10.1016/j.bmcl.2018.01.049 BindingDB Entry DOI: 10.7270/Q25T3P2R | |||||||||||
More data for this Ligand-Target Pair |