Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Apelin receptor (Homo sapiens (Human)) | BDBM269513 (N-(4-(2,6-dimethoxyphenyl)-5-(6-methyl-2-pyridinyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 830 | n/a | n/a | 7.5 | n/a |
AMGEN INC. US Patent | Assay Description The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV¿-3 expression vector (Si... | US Patent US10058550 (2018) BindingDB Entry DOI: 10.7270/Q26T0PP0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apelin receptor (Homo sapiens (Human)) | BDBM269513 (N-(4-(2,6-dimethoxyphenyl)-5-(6-methyl-2-pyridinyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 830 | n/a | n/a | n/a | n/a |
AMGEN INC. US Patent | Assay Description The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig... | US Patent US9845310 (2017) BindingDB Entry DOI: 10.7270/Q28P62TV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Apelin receptor (Homo sapiens (Human)) | BDBM269513 (N-(4-(2,6-dimethoxyphenyl)-5-(6-methyl-2-pyridinyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 830 | n/a | n/a | n/a | n/a |
AMGEN INC. US Patent | Assay Description The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV™-3 expression vector (Si... | US Patent US10221162 (2019) BindingDB Entry DOI: 10.7270/Q2ZK5JXS | |||||||||||
More data for this Ligand-Target Pair |